2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. Calcium Channel
  4. Gabapentin-d4

Gabapentin-d4 is the deuterium labeled Gabapentin. Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.

For research use only. We do not sell to patients.

Gabapentin-d<sub>4</sub> Chemical Structure

Gabapentin-d4 Chemical Structure

CAS No. : 1185039-20-6

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1 mg USD 260 In-stock
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Based on 1 publication(s) in Google Scholar

Other Forms of Gabapentin-d4:

Gabapentin-d4 Related Antibodies

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N-type calcium channel L-type calcium channel P/Q-type calcium channel T-type calcium channel Calcium Channel

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Description

Gabapentin-d4 is the deuterium labeled Gabapentin. Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Gabapentin-d4 Related Antibodies
Molecular Weight

175.26

Formula

C9H13D4NO2
CAS No.
Unlabeled CAS

60142-96-3
Appearance

Solid

Color

White to off-white

SMILES

OC(C([2H])([2H])C1(CCCCC1)C([2H])([2H])N)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

PBS : ≥ 10 mg/mL (57.06 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 5.7058 mL 28.5290 mL 57.0581 mL
5 mM 1.1412 mL 5.7058 mL 11.4116 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Concentration (final)

C2

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V2

In Vivo Dissolution Calculator
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Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
PBS 1 mM 5.7058 mL 28.5290 mL 57.0581 mL 142.6452 mL
5 mM 1.1412 mL 5.7058 mL 11.4116 mL 28.5290 mL
10 mM 0.5706 mL 2.8529 mL 5.7058 mL 14.2645 mL
15 mM 0.3804 mL 1.9019 mL 3.8039 mL 9.5097 mL
20 mM 0.2853 mL 1.4265 mL 2.8529 mL 7.1323 mL
25 mM 0.2282 mL 1.1412 mL 2.2823 mL 5.7058 mL
30 mM 0.1902 mL 0.9510 mL 1.9019 mL 4.7548 mL
40 mM 0.1426 mL 0.7132 mL 1.4265 mL 3.5661 mL
50 mM 0.1141 mL 0.5706 mL 1.1412 mL 2.8529 mL
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Gabapentin-d4 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Gabapentin-d41185039-20-6Calcium ChannelCa2+ channelsCa channelsInhibitorinhibitorinhibit

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