2. GPCR/G Protein
  3. GHSR
  4. Ghrelin receptor full agonist-2

Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.

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Ghrelin receptor full agonist-2 Chemical Structure

Ghrelin receptor full agonist-2 Chemical Structure

CAS No. : 2602452-73-1

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Ghrelin receptor full agonist-2 Related Antibodies

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Description

Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.

Cellular Effect
Cell Line Type Value Description References
HEK293 EC50
0.442 nM
Compound: 12j
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
HEK293 EC50
0.9 nM
Compound: 12j
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
[PMID: 32787075]
Molecular Weight

558.05

Formula

C26H28ClN5O5S
CAS No.
SMILES

O=C(C1=NOC(C2=C(C=CC=C2)Cl)=C1)N[C@@H]3[C@H](CN(C3)S(=O)(C4=CC=CC=C4)=O)C(N[C@H]5CCCNC5)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Ghrelin receptor full agonist-2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Ghrelin receptor full agonist-22602452-73-1Ghrelin receptor full agonist2Ghrelin receptor full agonist 2GHSRGrowth hormone secretagogue receptorGhrelin receptorInhibitorinhibitorinhibit

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Ghrelin receptor full agonist-2
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HY-145364
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