2. GPCR/G Protein
  3. GPR109A
  4. GPR81 agonist 2

GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 µM for hGPR81, hGPR109A, respectively.

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GPR81 agonist 2 Chemical Structure

GPR81 agonist 2 Chemical Structure

CAS No. : 1143024-28-5

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GPR81 agonist 2 Related Antibodies

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Description

GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 µM for hGPR81, hGPR109A, respectively[1].

IC50 & Target

EC50: 0.023 (hGPR81); 0.123 µM (hGPR109A)[1]
Molecular Weight

603.11

Formula

C26H27ClN6O5S2
CAS No.
SMILES

O=C(NC1=NC2=C(S1)C=C(S(=O)(C3CCN(CC3)C)=O)C=C2)NC(C4=C(Cl)C=C(OCC)C(N5N=CC=C5)=C4)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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GPR81 agonist 2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR81 agonist 21143024-28-5GPR109AHM74APUMA-GHCA2HCAR2 Inhibitorinhibitorinhibit

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GPR81 agonist 2
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HY-148563
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