2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. GR125487 sulfamate

GR125487 sulfamate is an orally active and selective antagonist of 5-HT4R. GR125487 sulfamate effectively blocks the cognition enhancing effect. GR125487 sulfamate can be used to study memory disorders, gastrointestinal disorders, mood disorders and urinary tract dysfunction.

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GR125487 sulfamate Chemical Structure

GR125487 sulfamate Chemical Structure

CAS No. : 859502-43-5

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GR125487 sulfamate Related Antibodies

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Description

GR125487 sulfamate is an orally active and selective antagonist of 5-HT4R. GR125487 sulfamate effectively blocks the cognition enhancing effect. GR125487 sulfamate can be used to study memory disorders, gastrointestinal disorders, mood disorders and urinary tract dysfunction[1].

Molecular Weight

524.58

Formula

C19H29FN4O8S2
CAS No.
SMILES

O=C(C1=C(NC2=C1C=C(F)C=C2)OC)OCC3CCN(CC3)CCNS(=O)(C)=O.O=S(O)(N)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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GR125487 sulfamate Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GR125487 sulfamate859502-43-55-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptor5-HT4RGR 125487Alzheimer’s diseaseAnimal models of cognitionInhibitorinhibitorinhibit

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