2. GPCR/G Protein
  3. GHSR
  4. K-(D-1-Nal)-FwLL-NH2 TFA

K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.

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K-(D-1-Nal)-FwLL-NH2 TFA Chemical Structure

K-(D-1-Nal)-FwLL-NH2 TFA Chemical Structure

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Other Forms of K-(D-1-Nal)-FwLL-NH2 TFA:

K-(D-1-Nal)-FwLL-NH2 TFA Related Antibodies

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Description

K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.

Molecular Weight

1016.16

Formula

C53H68F3N9O8
Sequence

Lys-{Nal}-Phe-Trp-Leu-Leu-NH2
Sequence Shortening

K{Nal}FWLL-NH2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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K-(D-1-Nal)-FwLL-NH2 TFA Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

K-(D-1-Nal)-FwLL-NH2GHSRGrowth hormone secretagogue receptorGhrelin receptorInhibitorinhibitorinhibit

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