2. GPCR/G Protein MAPK/ERK Pathway
  3. Ras
  4. KRAS G12C inhibitor 54

KRAS G12C inhibitor 54 (Compound 1) is a KRAS G12C inhibitor.

For research use only. We do not sell to patients.

KRAS G12C inhibitor 54 Chemical Structure

KRAS G12C inhibitor 54 Chemical Structure

CAS No. : 2765580-17-2

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KRAS G12C inhibitor 54 Related Antibodies

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Description

KRAS G12C inhibitor 54 (Compound 1) is a KRAS G12C inhibitor[1].

IC50 & Target

KRAS(G12C)

 

In Vitro

KRAS G12C inhibitor 54 (Compound 1) shows antiproliferative activity with an IC50 of 4.85 nM against H358 cells[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

KRAS G12C inhibitor 54 Related Antibodies
Molecular Weight

707.81

Formula

C36H40F3N7O3S
CAS No.
SMILES

C=CC(N1CC2(C1)CCN(CC2)C3=NC(N=S4(CCCCC4)=O)=NC5=C(C(C6=C7C=NNC7=CC=C6C)=C(C=C35)C8CC8)OCC(F)(F)F)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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KRAS G12C inhibitor 54 Related Classifications

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This equation is commonly abbreviated as: C1V1 = C2V2

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

KRAS G12C inhibitor 542765580-17-2RasantitumorH358Inhibitorinhibitorinhibit

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KRAS G12C inhibitor 54
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