LEI-101 free base

Cat. No.: HY-124283: FAQs
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LEI-101 free base is a selective and orally bioavailable CB2 receptor agonist with the potential to inhibit diseases associated with inflammation and/or oxidative stress. LEI-101 free base has a binding potency to CB2 receptors that is approximately 100 times higher than that to CB1 receptors. Its pEC50 value on CB2 receptors is 8, while its pKi value on hERG is less than 4. LEI-101 may have an inhibitory effect on conditions such as kidney disease.

For research use only. We do not sell to patients.

LEI-101 free base Chemical Structure

CAS No. : 1228660-00-1

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Other Forms of LEI-101 free base:

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Description	LEI-101 free base is a selective and orally bioavailable CB2 receptor agonist with the potential to inhibit diseases associated with inflammation and/or oxidative stress. LEI-101 free base has a binding potency to CB2 receptors that is approximately 100 times higher than that to CB1 receptors. Its pEC50 value on CB2 receptors is 8, while its pKi value on hERG is less than 4. LEI-101 may have an inhibitory effect on conditions such as kidney disease^[1].
Molecular Weight	472.53
Formula	C₂₃H₂₅FN₄O₄S
CAS No.	1228660-00-1
SMILES	O=C1N(C(CN1CC2=CC=C(C=C2)C3=NC(CN(CC4)CCS4(=O)=O)=C(C=C3)F)=O)C5CC5
Shipping	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation	Data Sheet (264 KB) Handling Instructions (2659 KB)
References	[1]. The novel, orally available and peripherally restricted selective cannabinoid CB2 receptor agonist LEI-101 prevents cisplatin-induced nephrotoxicity

LEI-101 free base Related Classifications

Inflammation/Immunology

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Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

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Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LEI-1011228660-00-1LEI101LEI 101Endogenous MetaboliteInhibitorinhibitorinhibit

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LEI-101 free base

Other Forms of LEI-101 free base:

LEI-101 free base Related Antibodies

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