2. Academic Validation
  3. Synthesis of a substance P antagonist with a somatostatin scaffold: factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry

Synthesis of a substance P antagonist with a somatostatin scaffold: factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry

  • J Med Chem. 2000 Oct 19;43(21):3827-31. doi: 10.1021/jm000316h.
J Liu 1,  D J Underwood,  M A Cascieri,  S P Rohrer,  L D Cantin,  G Chicchi,  A B Smith 3rd,  R Hirschmann
Affiliations

Affiliation

  • 1 Department of Chemistry, University of Pennsylvania, Philadelphia, Pennsylvania 19104, USA.
PMID: 11052787 DOI: 10.1021/jm000316h
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