2. GPCR/G Protein Neuronal Signaling
  3. Neurotensin Receptor
  4. MD01-67

MD01-67 is a selective macrocyclic compound targeting the neurotensin receptor type 2 (NTS2), with Ki of 2.9 nM. MD01-67 exhibits analgesic and tactile hypersensitivity reducing activity in rats acute/persistent/chronic inflammatory pain models.

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MD01-67 Chemical Structure

MD01-67 Chemical Structure

CAS No. : 2468971-42-6

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MD01-67 Related Antibodies

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Description

MD01-67 is a selective macrocyclic compound targeting the neurotensin receptor type 2 (NTS2), with Ki of 2.9 nM. MD01-67 exhibits analgesic and tactile hypersensitivity reducing activity in rats acute/persistent/chronic inflammatory pain models[1].

Molecular Weight

742.91

Formula

C37H58N8O8
CAS No.
SMILES

OC(C=C1)=CC=C1C[C@H](NC([C@H]2NC([C@@H](NC([C@@H](NC([C@H](C/C=C/C2)N)=O)CCCCN)=O)CCCCN)=O)=O)C(N[C@H](C(O)=O)CC3CCCC3)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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MD01-67 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MD01-672468971-42-6Neurotensin ReceptorSprague-Dawley ratanalgesictactile hypersensitivityInhibitorinhibitorinhibit

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