2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. MDA7

MDA7 is the selective agonist for cannabinoid receptor 2 with EC50 of 128 nM and 67.4 nM in human CB2 receptor and rat CB2 receptor. MDA7 exhibits good affinity to human CB2 receptor and rat CB2 receptor with Ki of 422 nM and 238 nM. MDA7 exhibits analgesic activity in rats models.

For research use only. We do not sell to patients.

MDA7 Chemical Structure

MDA7 Chemical Structure

CAS No. : 1103840-28-3

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MDA7 Related Antibodies

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Description

MDA7 is the selective agonist for cannabinoid receptor 2 with EC50 of 128 nM and 67.4 nM in human CB2 receptor and rat CB2 receptor. MDA7 exhibits good affinity to human CB2 receptor and rat CB2 receptor with Ki of 422 nM and 238 nM. MDA7 exhibits analgesic activity in rats models[1].

IC50 & Target

rat CB2-R

67.4 nM (IC50)

hCB2-R

128 nM (IC50)

rat CB2-R

238 nM (Ki)

hCB2-R

422 nM (Ki)

rCB1-R

2565 nM (Ki)

Molecular Weight

335.44

Formula

C22H25NO2
CAS No.
SMILES

O=C(N1CCCCC1)C2=CC=C3C(OCC3(CC4=CC=CC=C4)C)=C2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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MDA7 Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MDA71103840-28-3MDA 7MDA-7Cannabinoid ReceptorselectiveanalgesicratInhibitorinhibitorinhibit

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