1. GPCR/G Protein
  2. P2Y Receptor
  3. MRS2603

MRS2603 is a pyridoxal derivative. MRS2603 antagonized both P2Y1 and P2Y13 receptors.

For research use only. We do not sell to patients.

MRS2603 Chemical Structure

MRS2603 Chemical Structure

CAS No. : 860623-35-4

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Description

MRS2603 is a pyridoxal derivative. MRS2603 antagonized both P2Y1 and P2Y13 receptors[1].

IC50 & Target

P2Y1 Receptor

 

P2Y13 Receptor

 

In Vitro

MRS2603 inhibits phospholipase C (PLC) responses to 30 nM 2-methylthio-ADP (HY-108648A) in human P2Y1 receptor-mediated 1321N1 astrocytoma cells, with an IC50 of 0.245 μM[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

430.69

Formula

C14H12ClN4O8P

CAS No.
SMILES

O=CC1=C(COP(O)(O)=O)C(/N=N/C2=CC=C(Cl)C([N+]([O-])=O)=C2)=NC(C)=C1O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
MRS2603
Cat. No.:
HY-123202
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