2. GPCR/G Protein
  3. Adenosine Receptor
  4. N 0861

N-0861 is a novel selective A1 adenosine receptor antagonist. In studies, it has been shown to be able to inhibit the negative conduction effects (prolonged AH interval) and chest pain caused by adenosine, while having no significant effect on the increase in coronary blood flow velocity caused by adenosine. This indicates that N-0861 has the property of selectively inhibiting A1 adenosine receptors.

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N 0861 Chemical Structure

N 0861 Chemical Structure

CAS No. : 141696-90-4

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N 0861 Related Antibodies

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Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

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Description

N-0861 is a novel selective A1 adenosine receptor antagonist. In studies, it has been shown to be able to inhibit the negative conduction effects (prolonged AH interval) and chest pain caused by adenosine, while having no significant effect on the increase in coronary blood flow velocity caused by adenosine. This indicates that N-0861 has the property of selectively inhibiting A1 adenosine receptors[1].

Molecular Weight

243.31

Formula

C13H17N5
CAS No.
SMILES

CN(C=N1)C2=C1C(N[C@H]3[C@@H]4C[C@@H](CC4)C3)=NC=N2
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N 0861 Related Classifications

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Keywords:

N 0861141696-90-4N0861N-0861Adenosine ReceptorP1 receptorInhibitorinhibitorinhibit

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