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  3. NVS MLLT-1

NVS MLLT-1 (compound 3) is a potent and selective MLLT1 inhibitor with Kd values of 0.18 µM, 0.24 µM, and 0.22 µM for wild-type, T1 mutants, and T3 mutants, respectively.

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NVS MLLT-1 Chemical Structure

NVS MLLT-1 Chemical Structure

CAS No. : 2561471-13-2

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Based on 1 publication(s) in Google Scholar

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Description

NVS MLLT-1 (compound 3) is a potent and selective MLLT1 inhibitor with Kd values of 0.18 µM, 0.24 µM, and 0.22 µM for wild-type, T1 mutants, and T3 mutants, respectively[1][2].

IC50 & Target

Kd: 0.18 µM (wild-type); Kd: 0.24 µM (T1 mutants); Kd: 0.22 µM (T3 mutants)[1]

Molecular Weight

385.46

Formula

C23H23N5O

CAS No.
SMILES

O=C(C1=CC2=C(C=NC=C2)C=C1)NC3=CC=C4C(NC(CN5[C@H](CCC5)C)=N4)=C3

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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NVS MLLT-1
Cat. No.:
HY-160287
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