2. PROTAC
  3. Ligands for Target Protein for PROTAC
  4. OICR-9429-N-C2-NH2

OICR-9429-N-C2-NH2 is a ligand for Wd40 repeat domain protein 5 (WDR5) extracted from patent WO2019246570A1, intermediate 2. OICR-9429-N-C2-NH2 can be used in the synthesis of PROTACs.

For research use only. We do not sell to patients.

OICR-9429-N-C2-NH2 Chemical Structure

OICR-9429-N-C2-NH2 Chemical Structure

CAS No. : 2407457-55-8

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Based on 1 publication(s) in Google Scholar

OICR-9429-N-C2-NH2 Related Antibodies

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Description

OICR-9429-N-C2-NH2 is a ligand for Wd40 repeat domain protein 5 (WDR5) extracted from patent WO2019246570A1, intermediate 2. OICR-9429-N-C2-NH2 can be used in the synthesis of PROTACs[1].

IC50 & Target

Ligand for Target Protein for PROTAC[1]
In Vitro

PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

OICR-9429-N-C2-NH2 Related Antibodies
Molecular Weight

597.67

Formula

C31H38F3N7O2
CAS No.
SMILES

CN(CC1)CCN1C(C(NC(C2=CNC(C=C2C(F)(F)F)=O)=O)=C3)=CC=C3C4=CC(CN5CCN(CCN)CC5)=CC=C4
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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OICR-9429-N-C2-NH2 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

OICR-9429-N-C2-NH22407457-55-8Ligands for Target Protein for PROTACTarget Protein-binding MoietyWd40repeatdomainWDR5PROTACInhibitorinhibitorinhibit

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HY-141798
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