2. GPCR/G Protein
  3. Adenosine Receptor
  4. PD81723

PD81723 is an adenosine receptor binding enhancer. PD81723 enhances the inhibition of exogenous adenosine in a dose-dependent manner in hippocampal brain sections.

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PD81723 Chemical Structure

PD81723 Chemical Structure

CAS No. : 132861-87-1

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PD81723 Related Antibodies

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Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

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Description

PD81723 is an adenosine receptor binding enhancer. PD81723 enhances the inhibition of exogenous adenosine in a dose-dependent manner in hippocampal brain sections[1].

Cellular Effect
Cell Line Type Value Description References
CHO EC50
1.7 μM
Compound: PD-81723
Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells by scintillation counting
Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells by scintillation counting
[PMID: 20345101]
CHO-K1 ED50
13.6 μM
Compound: 1, PD-81723
Activity at human adenosine A1 receptor expressed in CHOK1 cells assessed as agonist-receptor ternary complex remaining by [35S]GTPgammaS binding assay
Activity at human adenosine A1 receptor expressed in CHOK1 cells assessed as agonist-receptor ternary complex remaining by [35S]GTPgammaS binding assay
[PMID: 17980606]
Molecular Weight

299.31

Formula

C14H12F3NOS
CAS No.
SMILES

O=C(C1=C(N)SC(C)=C1C)C2=CC=CC(C(F)(F)F)=C2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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PD81723 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PD81723132861-87-1PD 81723PD-81723Adenosine ReceptorP1 receptorAdenosine receptorReceptor modulatorHippocampal sliceInhibitorinhibitorinhibit

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