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  4. (R,R,S)-GAT107

(R,R,S)-GAT107 is a fully agonistic positive modulator of α7 nicotinic receptors with significant biological activity. Its activity is entirely present in its (+)-isomer 1b, while (-)-isomer 1a does not affect its activity when used together. Studies have shown that (R,R,S)-GAT107 is the most potent ago-PAM for α7 nicotinic receptors currently known and has the potential for further in vivo evaluation.

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(R,R,S)-GAT107 Chemical Structure

(R,R,S)-GAT107 Chemical Structure

CAS No. : 1426240-47-2

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(R,R,S)-GAT107 Related Antibodies

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Description

(R,R,S)-GAT107 is a fully agonistic positive modulator of α7 nicotinic receptors with significant biological activity. Its activity is entirely present in its (+)-isomer 1b, while (-)-isomer 1a does not affect its activity when used together. Studies have shown that (R,R,S)-GAT107 is the most potent ago-PAM for α7 nicotinic receptors currently known and has the potential for further in vivo evaluation[1].

Molecular Weight

405.31

Formula

C18H17BrN2O2S
CAS No.
SMILES

NS(=O)(C1=CC=C2N[C@@H](C3=CC=C(C=C3)Br)[C@](CC=C4)([H])[C@]4([H])C2=C1)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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(R,R,S)-GAT107 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(R,R,S)-GAT1071426240-47-2OthersInhibitorinhibitorinhibit

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