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Results for "

5'-Guanidinonaltrindole

" in MedChemExpress (MCE) Product Catalog:
Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-107748
    5'-Guanidinonaltrindole hydrochloride

    5'-GNTI hydrochloride

    		 Opioid Receptor Neurological Disease
    5'-Guanidinonaltrindole (5'-GNTI) hydrochloride is a highly selective and potent κ-opioid receptor antagonist with a Ki of 0.18 nM for human κ-opioid receptor .
    5'-Guanidinonaltrindole hydrochloride
  • HY-107748A
    5'-Guanidinonaltrindole TFA

    5'-GNTI TFA

    		 Others Neurological Disease
    5'-Guanidinonaltrindole TFA is a selective kappa-opioid receptor antagonist with significant opioid antagonist activity. 5'-Guanidinonaltrindole TFA exhibits 5 times the antagonistic potency of the prototypical kappa-opioid receptor antagonist norbinatorphimine in smooth muscle preparations, with a selectivity ratio exceeding 500 times. Binding and functional studies of 5'-Guanidinonaltrindole TFA showed pA(2) values comparable to smooth muscle data. 5'-Guanidinonaltrindole TFA is regarded as a potentially valuable pharmacological tool for studying opioids due to its high selectivity and potency .
    5'-Guanidinonaltrindole TFA

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