2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. VUF 5681 dihydrobromide

VUF 5681 dihydrobromide is a neutral antagonist of histamine H3 receptor. VUF 5681 dihydrobromide also has partial agonist function of H3 receptor. VUF 5681 dihydrobromide blocks the effects of Thioperamide (HY-12206). VUF 5681 dihydrobromide is used in central nervous system disease research.

For research use only. We do not sell to patients.

VUF 5681 dihydrobromide Chemical Structure

VUF 5681 dihydrobromide Chemical Structure

CAS No. : 639089-06-8

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VUF 5681 dihydrobromide Related Antibodies

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Description

VUF 5681 dihydrobromide is a neutral antagonist of histamine H3 receptor. VUF 5681 dihydrobromide also has partial agonist function of H3 receptor. VUF 5681 dihydrobromide blocks the effects of Thioperamide (HY-12206). VUF 5681 dihydrobromide is used in central nervous system disease research[1][2].

IC50 & Target

H3 receptor

 

In Vitro

VUF 5681 dihydrobromide (10 μM) blocks the stimulation of thioperamide in brain tissue[1].
VUF 5681 dihydrobromide (100 nM) inhibits other agonists in CHO-H3-SPAP cells[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

VUF 5681 dihydrobromide Related Antibodies
Molecular Weight

355.11

Formula

C11H21Br2N3
CAS No.
SMILES

C1(CCCC2CCNCC2)=CN=CN1.Br.Br
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Purity & Documentation
References
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VUF 5681 dihydrobromide Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

VUF 5681 dihydrobromide639089-06-8Histamine ReceptorNeutral antagonistHistamine H3 receptorsNeurological Disease，CHO-H3-SPAPInhibitorinhibitorinhibit

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