2. Metabolic Enzyme/Protease Neuronal Signaling GPCR/G Protein
  3. Aminopeptidase mGluR
  4. ZJ43

ZJ43 is a potent NAAG peptidase inhibitor, with an IC50 of 2.4 nM and a Ki of 0.8 nM. ZJ43 sufficiently activates group II mGluR and reduces some of the behavioral effects of PCP. ZJ43 shows an analgesic effect in neuropathic and inflammatory and pain models.

For research use only. We do not sell to patients.

ZJ43 Chemical Structure

ZJ43 Chemical Structure

CAS No. : 723331-20-2

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Based on 1 publication(s) in Google Scholar

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Description

ZJ43 is a potent NAAG peptidase inhibitor, with an IC50 of 2.4 nM and a Ki of 0.8 nM. ZJ43 sufficiently activates group II mGluR and reduces some of the behavioral effects of PCP. ZJ43 shows an analgesic effect in neuropathic and inflammatory and pain models[1].

IC50 & Target

IC50: 2.4 nM (NAAG)[1]
Molecular Weight

304.30

Formula

C12H20N2O7
CAS No.
SMILES

O=C(N[C@H](C(O)=O)CCC(O)=O)N[C@H](C(O)=O)CC(C)C
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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ZJ43 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ZJ43723331-20-2ZJ 43ZJ-43AminopeptidasemGluRMetabotropic glutamate receptorsAnalgesic effectNeuropathicInflammatoryInhibitorinhibitorinhibit

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