2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. GABA Receptor
  4. α5-GABAA receptor modulator 1

α5-GABAA receptor modulator 1 (Compound A-4) is a silencing allosteric modulator (SAM) specifically targeting the a5 subunit of the GABAA receptor, suitable for research into central nervous system (CNS) disorders.

For research use only. We do not sell to patients.

α5-GABAA receptor modulator 1 Chemical Structure

α5-GABAA receptor modulator 1 Chemical Structure

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α5-GABAA receptor modulator 1 Related Antibodies

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Description

α5-GABAA receptor modulator 1 (Compound A-4) is a silencing allosteric modulator (SAM) specifically targeting the a5 subunit of the GABAA receptor, suitable for research into central nervous system (CNS) disorders[1].

Molecular Weight

397.40

Formula

C21H20FN3O4
SMILES

CC1=C(C(C2=CC=C(C=C2)F)=NO1)COC3=CC4=C(C(N(CC4)CCO)=O)C=N3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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α5-GABAA receptor modulator 1 Related Classifications

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

α5-GABAA receptor modulator 1GABA ReceptorGamma-aminobutyric acid Receptorγ-Aminobutyric acid Receptorcentral nervous system (CNS)Inhibitorinhibitorinhibit

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