2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Monoamine Oxidase
  4. 5-HT6R/MAO-B modulator 1

5-HT6R/MAO-B modulator 1 (compound 48) is an antagonist of 5-HT6R at Gs signaling and an irreversible MAO-B inhibitor. 5-HT6R/MAO-B modulator 1 exhibits glioprotective properties. 5-HT6R/MAO-B modulator 1 can reverse Scopolamine-induced memory deficits. 5-HT6R/MAO-B modulator 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

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5-HT6R/MAO-B modulator 1 Chemical Structure

5-HT6R/MAO-B modulator 1 Chemical Structure

CAS No. : 2986222-45-9

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5-HT6R/MAO-B modulator 1 Related Antibodies

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MAO-A MAO-B

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Description

5-HT6R/MAO-B modulator 1 (compound 48) is an antagonist of 5-HT6R at Gs signaling and an irreversible MAO-B inhibitor. 5-HT6R/MAO-B modulator 1 exhibits glioprotective properties. 5-HT6R/MAO-B modulator 1 can reverse Scopolamine-induced memory deficits[1]. 5-HT6R/MAO-B modulator 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

IC50 & Target[1]

5-HT6 Receptor

 

MAO-B

 

Molecular Weight

584.77

Formula

C34H40N4O3S
CAS No.
SMILES

CN(CC#C)CC1=CC=C(C=C1)OCCCCCN2CCN(CC2)C3=C4C=CN(C4=CC=C3)S(=O)(C5=CC=CC=C5)=O
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Room temperature in continental US; may vary elsewhere.
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Purity & Documentation
References
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5-HT6R/MAO-B modulator 1 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

5-HT6R/MAO-B modulator 12986222-45-95-HT ReceptorMonoamine OxidaseSerotonin Receptor5-hydroxytryptamine ReceptorMAOglioprotectivescopolaminememory deficitsInhibitorinhibitorinhibit

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