2. Signaling Pathways
  3. GPCR/G Protein
  4. Protease Activated Receptor (PAR)
  5. PAR2 Isoform
  6. PAR2 Inhibitor

PAR2 Inhibitor

PAR2 Inhibitors (5):

Cat. No. Product Name Effect Purity
  • HY-120261
    GB-88
    		Inhibitor 99.05%
    GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.
  • HY-P1260
    FSLLRY-NH2
    		Inhibitor 98.52%
    FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.
  • HY-P1260A
    FSLLRY-NH2 TFA
    		Inhibitor 99.43%
    FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor.
  • HY-138558
    PAR-2-IN-1
    		Inhibitor 99.79%
    PAR-2-IN-1 is a protease-activated receptor-2 (PAR2) signaling pathway inhibitor with anti-inflammatory and anticancer effects.
  • HY-148016
    I-287
    		Inhibitor 99.36%
    I-287 is a orally active selective PAR2 inhibitor that acting as a negative allosteric regulator on Gαq and Gα12/13 activity and their downstream effectors. I-287 reduces Complete Freund's adjuvant (HY-153808)-induced inflammation in mice and can be used for inflammation/immunology research.