RAR/RXR Inhibitors

RXR β, EC₅₀: 400 nM

RXR γ, EC₅₀: 30 nM

RXR α

RXR α, EC₅₀: 2.1 μM

RXRγ, EC₅₀: 4.6 μM

RXR α

RXRβ

RXRγ

RXR α, Ki: 1.9 μM

RXR β, Ki: 0.64 μM

RXR γ, Ki: 1 μM

RXR α, Kd: 2 nM

RXR β, Kd: 2 nM

RXR γ, Kd: 2 nM

RXR α