1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. Src
  4. Src Inhibitors

Src Inhibitors

Lck

Fyn

Blk

Hck

Lyn

Yes

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Src Inhibitors
Product Name Lck Fyn Blk Hck Lyn Yes Purity
PRT062607 Hydrochloride
Lck, IC50: 249 nM ([2])
          98.07%
M4205
Lck, IC50: 141 nM
          99.47%
GLPG3312
Lck, IC50: 385 nM
Fyn, IC50: 447 nM
Blk, IC50: 730 nM
Hck, IC50: 2511 nM
Lyn, IC50: 272 nM
Yes, IC50: 598 nM
98.25%
AZM475271
Lck, IC50: 0.03 μM
          99.85%
PRT062607 acetate
Lck, IC50: 249 nM ([2])
          99.83%
SB 220025
p56-Lck, IC50: 3.5 μM
          99.90%
RK-20448
Lck, IC50: 0.24 μM
Fyn, IC50: 2.03 μM
Blk, IC50: 0.37 μM
      99.38%
Lck-IN-2
Lck, IC50: 10.6 nM
         
BMS-243117
Lck, IC50: 4 nM
Fyn, IC50: 32 nM
Blk, IC50: 84 nM