BD-1008 dihydrobromide

Cat. No.: HY-100966 Purity: 98.07%: FAQs
Data Sheet SDS COA Handling Instructions Technical Support

BD-1008 dihydrobromide is an antagonist of sigma Receptor.

For research use only. We do not sell to patients.

BD-1008 dihydrobromide Chemical Structure

Size	Stock	Quantity
1 mg	In-stock	Estimated Time of Arrival: December 31
5 mg	In-stock	Estimated Time of Arrival: December 31
10 mg	In-stock	Estimated Time of Arrival: December 31
50 mg	Get quote
100 mg	Get quote

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Other Forms of BD-1008 dihydrobromide:

BD-1008-d₅ dihydrobromide Get quote
BD-1008 Get quote

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Biological Activity
Purity & Documentation
References
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Description

BD-1008 dihydrobromide is an antagonist of sigma Receptor^[1].

Molecular Weight

463.08

Formula

C₁₅H₂₄Br₂Cl₂N₂

CAS No.

138356-09-9

Appearance

Solid

Color

White to off-white

SMILES

CN(CCC1=CC=C(Cl)C(Cl)=C1)CCN2CCCC2.Br.Br

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

DMSO : 50 mg/mL (107.97 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.1595 mL	10.7973 mL	21.5945 mL
5 mM	0.4319 mL	2.1595 mL	4.3189 mL
10 mM	0.2159 mL	1.0797 mL	2.1595 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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In Vivo Dissolution Calculator

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 98.07%

Select Batch:

Data Sheet (267 KB) SDS (251 KB)

COA (246 KB) HNMR (284 KB) LCMS (88 KB)

Handling Instructions (2659 KB)

References

[1]. Matsumoto RR, et al. Novel analogs of the sigma receptor ligand BD1008 attenuate cocaine-induced toxicity in mice. Eur J Pharmacol. 2004 May 10;492(1):21-6. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.1595 mL	10.7973 mL	21.5945 mL	53.9864 mL
	5 mM	0.4319 mL	2.1595 mL	4.3189 mL	10.7973 mL
	10 mM	0.2159 mL	1.0797 mL	2.1595 mL	5.3986 mL
	15 mM	0.1440 mL	0.7198 mL	1.4396 mL	3.5991 mL
	20 mM	0.1080 mL	0.5399 mL	1.0797 mL	2.6993 mL
	25 mM	0.0864 mL	0.4319 mL	0.8638 mL	2.1595 mL
	30 mM	0.0720 mL	0.3599 mL	0.7198 mL	1.7995 mL
	40 mM	0.0540 mL	0.2699 mL	0.5399 mL	1.3497 mL
	50 mM	0.0432 mL	0.2159 mL	0.4319 mL	1.0797 mL
	60 mM	0.0360 mL	0.1800 mL	0.3599 mL	0.8998 mL
	80 mM	0.0270 mL	0.1350 mL	0.2699 mL	0.6748 mL
	100 mM	0.0216 mL	0.1080 mL	0.2159 mL	0.5399 mL