2. Neuronal Signaling
  3. AAK1
  4. BMT-124110 formic

BMT-124110 formic is a potent, selective AAK1 inhibitor, with an IC50 of 0.9 nM. BMT-124110 shows antinociceptive activity. BMT-124110 formic inhibits BMP-2-inducible protein kinase (BIKE) and Cyclin G-associated kinase (GAK) with IC50s of 17 and 99 nM, respectively.

For research use only. We do not sell to patients.

BMT-124110 formic Chemical Structure

BMT-124110 formic Chemical Structure

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Based on 1 publication(s) in Google Scholar

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Description

BMT-124110 formic is a potent, selective AAK1 inhibitor, with an IC50 of 0.9 nM. BMT-124110 shows antinociceptive activity. BMT-124110 formic inhibits BMP-2-inducible protein kinase (BIKE) and Cyclin G-associated kinase (GAK) with IC50s of 17 and 99 nM, respectively[1].

Molecular Weight

415.48

Formula

C22H29N3O5
Appearance

Solid

SMILES

CC(NC1=CC2=C(COC3=CC(OC[C@@](C)(N)CC(C)C)=CC=C32)C=N1)=O.OC=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Purity & Documentation
References
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BMT-124110 formic Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

BMT-124110BMT124110BMT 124110AAK1Adaptor-associated Kinase 1AP2-associated kinase 1neuropathicpainchronicconstrictioninjuryCCIBIKEGAKInhibitorinhibitorinhibit

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