2. Metabolic Enzyme/Protease
  3. CETP
  4. CETP-IN-3

CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively.

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CETP-IN-3 Chemical Structure

CETP-IN-3 Chemical Structure

CAS No. : 939391-31-8

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CETP-IN-3 Related Antibodies

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Description

CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].

Cellular Effect
Cell Line Type Value Description References
HEK293 IC50
> 80 μM
Compound: 13
Inhibition of human ERG expressed in HEK293 cells by whole cell patch clamp method
Inhibition of human ERG expressed in HEK293 cells by whole cell patch clamp method
[PMID: 31223447]
Molecular Weight

704.50

Formula

C30H24F12N2O4
CAS No.
SMILES

O=C(N[C@@](C1=CC(OC(F)(F)C(F)F)=CC(F)=C1)(C2=CC=C(F)C(OC3CC3)=C2)CC4=CC=CC=C4)C(N)C(C(F)(F)F)(O)C(F)(F)F
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Purity & Documentation
References
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CETP-IN-3 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CETP-IN-3939391-31-8CETPCholesteryl ester transfer proteinInhibitorinhibitorinhibit

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