2. Metabolic Enzyme/Protease Epigenetics Cell Cycle/DNA Damage
  3. Cytochrome P450 HDAC
  4. CYP17A1/HDAC6-IN-1

CYP17A1/HDAC6-IN-1 (compound 12) is a potent inhibitor of CYP17A1/HDAC6, with IC50 of 0.284μM and 0.6015 μM,respectively. CYP17A1/HDAC6-IN-1 has anti-tumor activity.

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CYP17A1/HDAC6-IN-1 Chemical Structure

CYP17A1/HDAC6-IN-1 Chemical Structure

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CYP17A1/HDAC6-IN-1 Related Antibodies

Top Publications Citing Use of Products

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CYP1 CYP2 CYP3 CYP4 CYP11 CYP17 Aromatase/CYP19A1 CYP26 CYP51 CYP1A2 CYP2D6 CYP2C9 CYP2C19 CYP3A4 CYP17A1

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View All Isoforms
HDAC HDAC1 HDAC2 HDAC3 HDAC4 HDAC5 HDAC6 HDAC7 HDAC8 HDAC9 HDAC10 HDAC11 HD1 HD2

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Description

CYP17A1/HDAC6-IN-1 (compound 12) is a potent inhibitor of CYP17A1/HDAC6, with IC50 of 0.284μM and 0.6015 μM,respectively. CYP17A1/HDAC6-IN-1 has anti-tumor activity[1].

IC50 & Target

CYP17A1

0.284 μM (IC50)

HDAC6

0.6015 μM (IC50)

Molecular Weight

506.68

Formula

C31H42N2O4
SMILES

C[C@]12CCC3C(CC=C4C[C@@H](OC(CCCCCC(NO)=O)=O)CC[C@@]43C)C1CC=C2C5=CN=CC=C5
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CYP17A1/HDAC6-IN-1 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CYP17A1/HDAC6-IN-1Cytochrome P450HDACCYPsHistone deacetylasesGBM cellsDNA damageInhibitorinhibitorinhibit

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