2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. Deltasonamide 2

Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.

At equivalent molar concentrations, both the salt and free forms of a compound exhibit comparable biological activity. Nevertheless, the salt form (Deltasonamide 2 (TFA) and Deltasonamide 2 hydrochloride) usually boasts enhanced water solubility and stability.

For research use only. We do not sell to patients.

Deltasonamide 2 Chemical Structure

Deltasonamide 2 Chemical Structure

CAS No. : 2088485-34-9

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Other Forms of Deltasonamide 2:

Deltasonamide 2 Related Antibodies

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PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

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Description

Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM[1].

IC50 & Target

Kd: ~385 pM (PDEδ)[1]
Cellular Effect
Cell Line Type Value Description References
AGS IC50
1.2 μM
Compound: Deltasonamide 2
Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
MIA PaCa-2 IC50
507 nM
Compound: Deltasonamide 2
Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
NCI-H358 IC50
954 nM
Compound: Deltasonamide 2
Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
PaTu 8988t IC50
1.2 μM
Compound: Deltasonamide 2
Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
Molecular Weight

647.25

Formula

C30H39ClN6O4S2
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=S(C1=CC=C(S(=O)(N(CC2=CC=C(Cl)C=C2)C3CCCC3)=O)C=C1)(N([C@H]4CC[C@H](N)CC4)CC5=NC(NC)=NC=C5)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Deltasonamide 2 Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Deltasonamide 22088485-34-9Deltasonamide2Deltasonamide-2Phosphodiesterase (PDE)Inhibitorinhibitorinhibit

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