2. GPCR/G Protein
  3. G protein-coupled Bile Acid Receptor 1 Leukotriene Receptor
  4. GPBAR1-IN-3

GPBAR1-IN-3 (Compound 14) is a selective GPBAR1 agonist (EC50=0.17 μM) and a CysLT1R antagonist.

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GPBAR1-IN-3 Chemical Structure

GPBAR1-IN-3 Chemical Structure

CAS No. : 2760546-05-0

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Description

GPBAR1-IN-3 (Compound 14) is a selective GPBAR1 agonist (EC50=0.17 μM) and a CysLT1R antagonist[1].

Molecular Weight

321.41

Formula

C21H23NO2
CAS No.
SMILES

CC(CC)COC1=CC(OCC2=NC3=C(C=C2)C=CC=C3)=CC=C1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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GPBAR1-IN-3 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

GPBAR1-IN-32760546-05-0G protein-coupled Bile Acid Receptor 1Leukotriene ReceptorG-protein coupled receptor 19GPCR19TGR5GPBAR1GPCRCysLT1RInhibitorinhibitorinhibit

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HY-145234
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