2. GPCR/G Protein Neuronal Signaling
  3. GPR55
  4. GPR55 agonist 3

GPR55 agonist 3 (Compound 26) is a GPR55 agonist (EC50: 0.239 nM, and 1.76 nM for hGPR55 and rGPR55). GPR55 agonist 3 induces β-arrestin recruitment to human GPR55 (EC50: 6.2 nM).

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GPR55 agonist 3 Chemical Structure

GPR55 agonist 3 Chemical Structure

CAS No. : 3006105-44-5

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GPR55 agonist 3 Related Antibodies

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Description

GPR55 agonist 3 (Compound 26) is a GPR55 agonist (EC50: 0.239 nM, and 1.76 nM for hGPR55 and rGPR55). GPR55 agonist 3 induces β-arrestin recruitment to human GPR55 (EC50: 6.2 nM)[1].

Molecular Weight

376.35

Formula

C19H16F4N4
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

FC(F)(F)CC1=CN=CC(C2=CN=C(N[C@@H](C3=CC=C(F)C=C3)C)C=N2)=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 250 mg/mL (664.28 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6571 mL 13.2855 mL 26.5710 mL
5 mM 0.5314 mL 2.6571 mL 5.3142 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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In Vivo Dissolution Calculator
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Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.6571 mL 13.2855 mL 26.5710 mL 66.4275 mL
5 mM 0.5314 mL 2.6571 mL 5.3142 mL 13.2855 mL
10 mM 0.2657 mL 1.3286 mL 2.6571 mL 6.6428 mL
15 mM 0.1771 mL 0.8857 mL 1.7714 mL 4.4285 mL
20 mM 0.1329 mL 0.6643 mL 1.3286 mL 3.3214 mL
25 mM 0.1063 mL 0.5314 mL 1.0628 mL 2.6571 mL
30 mM 0.0886 mL 0.4429 mL 0.8857 mL 2.2143 mL
40 mM 0.0664 mL 0.3321 mL 0.6643 mL 1.6607 mL
50 mM 0.0531 mL 0.2657 mL 0.5314 mL 1.3286 mL
60 mM 0.0443 mL 0.2214 mL 0.4429 mL 1.1071 mL
80 mM 0.0332 mL 0.1661 mL 0.3321 mL 0.8303 mL
100 mM 0.0266 mL 0.1329 mL 0.2657 mL 0.6643 mL
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GPR55 agonist 3 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR55 agonist 33006105-44-5GPR55G protein-coupled receptor 55β-arrestin recruitmentGPR55 activationInhibitorinhibitorinhibit

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