2. PI3K/Akt/mTOR
  3. PI3K
  4. LAS191954

LAS191954 is a potent, selective and orally active PI3Kδ inhibitor for inflammatory diseases treatment, with an IC50 of 2.6 nM.

For research use only. We do not sell to patients.

LAS191954 Chemical Structure

LAS191954 Chemical Structure

CAS No. : 1403947-26-1

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LAS191954 Related Antibodies

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PI3Kα PI3Kβ PI3Kγ PI3Kδ PI3KC2α PI3KC2β PI3KC2γ Vps34 PI3K PI3KC3 p120γ

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Description

LAS191954 is a potent, selective and orally active PI3Kδ inhibitor for inflammatory diseases treatment, with an IC50 of 2.6 nM[1].

IC50 & Target[1]

PI3Kδ

2.6 nM (IC50)

Molecular Weight

397.39

Formula

C20H15N9O
CAS No.
SMILES

O=C1N(C2=CC=CC=C2)C([C@@H](NC3=C(C#N)C(N)=NC=N3)C)=NN4C1=C(C#N)C=C4
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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LAS191954 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LAS1919541403947-26-1LAS 191954LAS-191954PI3KPhosphoinositide 3-kinaseInhibitorinhibitorinhibit

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LAS191954
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HY-101114
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