Norgestimate metabolite norelgestromin-d₆ (Synonyms: 17-Deacetyl norgestimate-d₆; 17-Deacylnorgestimate-d₆)

Cat. No.: HY-G0018S: FAQs
Data Sheet Handling Instructions

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Norgestimate metabolite norelgestromin-d₆ is the deuterium labeled Norgestimate metabolite norelgestromin. Norelgestromin is a metabolite of Norgestimate, which is a progestin or synthetic progestogen. Norgestimate metabolite norelgestromin-d6 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

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Norgestimate metabolite norelgestromin-d<sub>6</sub> Chemical Structure

Norgestimate metabolite norelgestromin-d₆ Chemical Structure

CAS No. : 1263184-13-9

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1 mg	USD 270	In-stock	Estimated Time of Arrival: December 31
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10 mg		Get quote

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Other Forms of Norgestimate metabolite norelgestromin-d₆:

Norgestimate metabolite Norelgestromin In-stock

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Description

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

333.50

Formula

C₂₁H₂₃D₆NO₂

CAS No.

1263184-13-9

Unlabeled CAS

53016-31-2

Appearance

Solid

Color

White to off-white

SMILES

CC[C@@]12[C@](CC[C@@]2(O)C#C)([H])[C@@]3([H])[C@]([C@]4([2H])C(C([2H])([2H])C3)=C([2H])/C(C([2H])([2H])C4)=N/O)([H])CC1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

DMSO : 20 mg/mL (59.97 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.9985 mL	14.9925 mL	29.9850 mL
5 mM	0.5997 mL	2.9985 mL	5.9970 mL
10 mM	0.2999 mL	1.4993 mL	2.9985 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

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mg/kg

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(per animal)

μL

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.9985 mL	14.9925 mL	29.9850 mL	74.9625 mL
	5 mM	0.5997 mL	2.9985 mL	5.9970 mL	14.9925 mL
	10 mM	0.2999 mL	1.4993 mL	2.9985 mL	7.4963 mL
	15 mM	0.1999 mL	0.9995 mL	1.9990 mL	4.9975 mL
	20 mM	0.1499 mL	0.7496 mL	1.4993 mL	3.7481 mL
	25 mM	0.1199 mL	0.5997 mL	1.1994 mL	2.9985 mL
	30 mM	0.1000 mL	0.4998 mL	0.9995 mL	2.4988 mL
	40 mM	0.0750 mL	0.3748 mL	0.7496 mL	1.8741 mL
	50 mM	0.0600 mL	0.2999 mL	0.5997 mL	1.4993 mL

Norgestimate metabolite norelgestromin-d₆ Related Classifications

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Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Norgestimate metabolite norelgestromin-d₆1263184-13-917-Deacetyl norgestimate-d₆17-Deacylnorgestimate-d₆Isotope-Labeled CompoundsDrug MetaboliteInhibitorinhibitorinhibit

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Norgestimate metabolite norelgestromin-d6 (Synonyms: 17-Deacetyl norgestimate-d6; 17-Deacylnorgestimate-d6)

Other Forms of Norgestimate metabolite norelgestromin-d6:

Norgestimate metabolite norelgestromin-d6 Related Antibodies