2. Membrane Transporter/Ion Channel Neuronal Signaling Metabolic Enzyme/Protease
  3. TRP Channel Endogenous Metabolite
  4. OMDM-5

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM).

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OMDM-5 Chemical Structure

OMDM-5 Chemical Structure

CAS No. : 616884-66-3

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Based on 1 publication(s) in Google Scholar

OMDM-5 Related Antibodies

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Description

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].

IC50 & Target

Ki: 4.8 μM (anandamide cellular uptake), 4.9 μM (CB1), EC50: 75 nM (VR1)[1]
Molecular Weight

432.64

Formula

C26H44N2O3
CAS No.
SMILES

CCCCCCCC/C=C\CCCCCCCC(NNCC1=CC=C(O)C(OC)=C1)=O
Structure Classification
Initial Source
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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OMDM-5 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

OMDM-5616884-66-3OMDM5OMDM 5TRP ChannelEndogenous MetaboliteTransient receptor potential channelsfattyacidsuptakeRBL-2H3cellsvanilloidVR1cannabinoidreceptortype1CB1CB2FAAHInhibitorinhibitorinhibit

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