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Results for "

farnesyl-protein transferase

" in MedChemExpress (MCE) Product Catalog:

6

Inhibitors & Agonists

1

Peptides

4

Natural
Products

Targets Recommended:
Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-N2150
    Psammaplin A

    		HDAC DNA Methyltransferase DNA/RNA Synthesis Bacterial Apoptosis Infection Inflammation/Immunology Cancer
    Psammaplin A is a marine metabolite. Psammaplin A is a selective HDAC1 inhibitor (IC50: 45 nM), an inhibitor of DNA methyltransferases (IC50: 18.6 nM), APN (IC50: 18 μM), DNA topoisomerase, farnesyl protein transferase, and leucine aminopeptidase. Psammaplin A is a PPARγ activator and induces apoptosis. Psammaplin A has antitumor and anti-inflammatory activities. Psammaplin A has antibacterial activity against Gram-positive bacteria and inhibits DNA synthesis and DNA gyrase activity. Psammaplin A inhibits angiogenesis. Psammaplin A can be used in cancer and bacterial research .
    Psammaplin A
  • HY-125311
    Zaragozic acid D

    		Farnesyl Transferase Cancer
    Zaragozic acid D is a squalene synthase inhibitor. Zaragozic acid D also is a farnesyl-protein transferase (FPTase) inhibitor with an IC50 value of 100 nM for bovine FPTase .
    Zaragozic acid D
  • HY-W022657
    H-Met-OiPr hydrochloride

    		Amino Acid Derivatives Others
    H-Met-OiPr hydrochloride is an Methionine derivative. H-Met-OiPr hydrochloride participates in the synthesis preparation of inhibitors of farnesyl-protein transferase (FTase), and can be used in cancer research .
    H-Met-OiPr hydrochloride
  • HY-126871
    Zaragozic acid D2

    		Farnesyl Transferase Metabolic Disease Cancer
    Zaragozic acid D2 is the inhibitor for squalene synthase and Ras farnesyl-protein transferase (Ras FPTase), with IC50 of 2 nM and 100 nM, respectively. Zaragozic acid D2 is potentially ameliorating hypercholesterolemia and Ras-induced cancer .
    Zaragozic acid D2
  • HY-134579
    Chaetomellic acid A

    		Farnesyl Transferase Inflammation/Immunology
    Chaetomellic acid A can be isolated from Chaetomella acutiseta. Chaetomellic acid A is a specific inhibitor of farnesyl-protein transferase. Chaetomellic acid A decreases oxidative stress-induced apoptosis in cells. Chaetomellic acid A reduces renal damage after unilateral ureteral obstruction (UUO) in mice .
    Chaetomellic acid A
  • HY-118426
    (Rac)-Tipifarnib

    (Rac)-IND 58359; (Rac)-R115777

    		 Farnesyl Transferase Ras Cancer
    (Rac)-Tipifarnib ((Rac)-IND 58359; (Rac)-R115777) is a potent farnesyl protein transferase inhibitor that specifically targets the pro-tailation process of Ras proteins. (Rac)-Tipifarnib showed significant in vivo antitumor effects after oral administration to mice .
    (Rac)-Tipifarnib

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