Sodium Channel inhibitor 4

Cat. No.: HY-49066 Purity: ≥98.0%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Sodium Channel inhibitor 4 is a sodium channel inhibitor.

For research use only. We do not sell to patients.

Sodium Channel inhibitor 4 Chemical Structure

CAS No. : 587843-16-1

Size	Price	Stock	Quantity
5 mg	USD 50	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 80	In-stock	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

or Bulk Inquiry

* Please select Quantity before adding items.

This product is a controlled substance and not for sale in your territory.

Customer Review

Based on 1 publication(s) in Google Scholar

Featured Recommendations

•Related Screening Libraries:

•Related Small Molecules:

•Related Proteins:

View All Sodium Channel Isoform Specific Products:

View All Isoforms

Na_v1.1 Na_v1.2 Na_v1.3 Na_v1.4 Na_v1.5 Na_v1.6 Na_v1.7 Na_v1.8

Biological Activity
Purity & Documentation
References
Customer Review

Description

Sodium Channel inhibitor 4 is a sodium channel inhibitor^[1].

Molecular Weight

451.95

Formula

C₁₉H₁₈ClN₃O₄S₂

CAS No.

587843-16-1

Appearance

Solid

Color

White to off-white

SMILES

CC(C)(OC1=CC=C(Cl)C=C1)C(NC2=CC=C(S(=O)(NC3=NC=CS3)=O)C=C2)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL (221.26 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.2126 mL	11.0632 mL	22.1263 mL
5 mM	0.4425 mL	2.2126 mL	4.4253 mL
10 mM	0.2213 mL	1.1063 mL	2.2126 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Molarity Calculator
Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: ≥98.0%

Select Batch:

Data Sheet (267 KB) SDS (251 KB)

COA (247 KB) HNMR (151 KB)

Handling Instructions (2659 KB)

References

[1]. Gonzalez, et al. Preparation of N-(4-sulfamoylphenyl) amides as inhibitors of voltage-gated sodium channels. United States, US20060025415 A1. 2006-02-02.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.2126 mL	11.0632 mL	22.1263 mL	55.3159 mL
	5 mM	0.4425 mL	2.2126 mL	4.4253 mL	11.0632 mL
	10 mM	0.2213 mL	1.1063 mL	2.2126 mL	5.5316 mL
	15 mM	0.1475 mL	0.7375 mL	1.4751 mL	3.6877 mL
	20 mM	0.1106 mL	0.5532 mL	1.1063 mL	2.7658 mL
	25 mM	0.0885 mL	0.4425 mL	0.8851 mL	2.2126 mL
	30 mM	0.0738 mL	0.3688 mL	0.7375 mL	1.8439 mL
	40 mM	0.0553 mL	0.2766 mL	0.5532 mL	1.3829 mL
	50 mM	0.0443 mL	0.2213 mL	0.4425 mL	1.1063 mL
	60 mM	0.0369 mL	0.1844 mL	0.3688 mL	0.9219 mL
	80 mM	0.0277 mL	0.1383 mL	0.2766 mL	0.6914 mL
	100 mM	0.0221 mL	0.1106 mL	0.2213 mL	0.5532 mL