2. Protein Tyrosine Kinase/RTK
  3. Src
  4. SRC-3-IN-2

SRC-3-IN-2 (SI-12 6c)is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity.

For research use only. We do not sell to patients.

SRC-3-IN-2 Chemical Structure

SRC-3-IN-2 Chemical Structure

CAS No. : 3074959-44-4

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SRC-3-IN-2 Related Antibodies

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Description

SRC-3-IN-2 (SI-12 6c)is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity[1].

In Vitro

SRC-3-IN-2 IC50 value of MCF7 cell is 3.4 nM[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

SRC-3-IN-2 Related Antibodies
In Vivo


Pharmacokinetic Analysis in CD-1 mice Model[1]

Route Dose (mg/kg) AUClast (ng·h/mL) t1/2 (h) Tmax (h) Cmax (ng/mL) Clobs (mL·min/kg) F (%)
i.v. 1 737 22.5 0.033 1066 22 /
p.o. 10 1719 14.3 0.25 217 / 24.6

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

319.28

Formula

C15H12F3N5
CAS No.
SMILES

CN1C2=CC(F)=C(F)C=C2N/C1=N\N=C(C3=CC=C(C=N3)F)/C
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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SRC-3-IN-2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SRC-3-IN-23074959-44-4SrcSRCInhibitorMCF7Antitumorinhibitorinhibit

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