2. Protein Tyrosine Kinase/RTK
  3. Src
  4. SRC-3-IN-2

SRC-3-IN-2 (SI-12 6c)is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity.

For research use only. We do not sell to patients.

SRC-3-IN-2 Chemical Structure

SRC-3-IN-2 Chemical Structure

CAS No. : 3074959-44-4

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SRC-3-IN-2 Related Antibodies

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Description

SRC-3-IN-2 (SI-12 6c)is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity[1].

In Vitro

SRC-3-IN-2 IC50 value of MCF7 cell is 3.4 nM[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

SRC-3-IN-2 Related Antibodies
In Vivo


Pharmacokinetic Analysis in CD-1 mice Model[1]

Route Dose (mg/kg) AUClast (ng·h/mL) t1/2 (h) Tmax (h) Cmax (ng/mL) Clobs (mL·min/kg) F (%)
i.v. 1 737 22.5 0.033 1066 22 /
p.o. 10 1719 14.3 0.25 217 / 24.6

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

319.28

Formula

C15H12F3N5
CAS No.
Appearance

Solid

Color

Purple to purplish red

SMILES

CN1C2=CC(F)=C(F)C=C2N/C1=N\N=C(C3=CC=C(C=N3)F)/C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Purity & Documentation
References
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SRC-3-IN-2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SRC-3-IN-23074959-44-4SrcSRCInhibitorMCF7Antitumorinhibitorinhibit

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HY-163469
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