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  3. Drug Derivative
  4. Tosylate-DPA-714

Tosylate-DPA-714 (compound 2) is a DPA-714 (HY-122607) tosylate analog. Tosylate-DPA-714 is a precursor for 18F-DPA-714. DPA-714 is a translocator protein (TSPO)-specific ligand.

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Tosylate-DPA-714 Chemical Structure

Tosylate-DPA-714 Chemical Structure

CAS No. : 958233-17-5

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Tosylate-DPA-714 Related Antibodies

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Description

Tosylate-DPA-714 (compound 2) is a DPA-714 (HY-122607) tosylate analog. Tosylate-DPA-714 is a precursor for 18F-DPA-714. DPA-714 is a translocator protein (TSPO)-specific ligand[1].

Molecular Weight

550.67

Formula

C29H34N4O5S
CAS No.
Appearance

Solid

SMILES

O=C(CC1=C(N=C(C)C=C2C)N2N=C1C3=CC=C(OCCOS(=O)(C4=CC=C(C)C=C4)=O)C=C3)N(CC)CC
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Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (181.60 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.8160 mL 9.0798 mL 18.1597 mL
5 mM 0.3632 mL 1.8160 mL 3.6319 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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In Vivo Dissolution Calculator
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Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 1.8160 mL 9.0798 mL 18.1597 mL 45.3992 mL
5 mM 0.3632 mL 1.8160 mL 3.6319 mL 9.0798 mL
10 mM 0.1816 mL 0.9080 mL 1.8160 mL 4.5399 mL
15 mM 0.1211 mL 0.6053 mL 1.2106 mL 3.0266 mL
20 mM 0.0908 mL 0.4540 mL 0.9080 mL 2.2700 mL
25 mM 0.0726 mL 0.3632 mL 0.7264 mL 1.8160 mL
30 mM 0.0605 mL 0.3027 mL 0.6053 mL 1.5133 mL
40 mM 0.0454 mL 0.2270 mL 0.4540 mL 1.1350 mL
50 mM 0.0363 mL 0.1816 mL 0.3632 mL 0.9080 mL
60 mM 0.0303 mL 0.1513 mL 0.3027 mL 0.7567 mL
80 mM 0.0227 mL 0.1135 mL 0.2270 mL 0.5675 mL
100 mM 0.0182 mL 0.0908 mL 0.1816 mL 0.4540 mL
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Tosylate-DPA-714 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Tosylate-DPA-714958233-17-5Drug DerivativeDrug derivative18F-fluorideDPA-714translocator proteinInhibitorinhibitorinhibit

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