2. Neuronal Signaling
  3. Sigma Receptor
  4. Trifluperidol hydrochloride

Trifluperidol hydrochloride  (Synonyms: R 2498)

Cat. No.: HY-124462 Purity: 99.4%
COA Handling Instructions

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Trifluperidol hydrochloride is a Sigma-1 receptor antagonist with a Ki value of 3.3 nM. Trifluperidol hydrochloride is used in the study of psychosis.

For research use only. We do not sell to patients.

Trifluperidol hydrochloride Chemical Structure

Trifluperidol hydrochloride Chemical Structure

CAS No. : 2062-77-3

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Trifluperidol hydrochloride Related Antibodies

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Description

Trifluperidol hydrochloride is a Sigma-1 receptor antagonist with a Ki value of 3.3 nM. Trifluperidol hydrochloride is used in the study of psychosis[1].

Molecular Weight

445.88

Formula

C22H24ClF4NO2
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(CCCN1CCC(O)(CC1)C2=CC=CC(C(F)(F)F)=C2)C3=CC=C(C=C3)F.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 40 mg/mL (89.71 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2428 mL 11.2138 mL 22.4276 mL
5 mM 0.4486 mL 2.2428 mL 4.4855 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 99.4%

COA (245 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.2428 mL 11.2138 mL 22.4276 mL 56.0689 mL
5 mM 0.4486 mL 2.2428 mL 4.4855 mL 11.2138 mL
10 mM 0.2243 mL 1.1214 mL 2.2428 mL 5.6069 mL
15 mM 0.1495 mL 0.7476 mL 1.4952 mL 3.7379 mL
20 mM 0.1121 mL 0.5607 mL 1.1214 mL 2.8034 mL
25 mM 0.0897 mL 0.4486 mL 0.8971 mL 2.2428 mL
30 mM 0.0748 mL 0.3738 mL 0.7476 mL 1.8690 mL
40 mM 0.0561 mL 0.2803 mL 0.5607 mL 1.4017 mL
50 mM 0.0449 mL 0.2243 mL 0.4486 mL 1.1214 mL
60 mM 0.0374 mL 0.1869 mL 0.3738 mL 0.9345 mL
80 mM 0.0280 mL 0.1402 mL 0.2803 mL 0.7009 mL
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Trifluperidol hydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Trifluperidol2062-77-3R 2498R2498R-2498Sigma ReceptorSigma-1 receptorAntagonistantipsychoticInhibitorinhibitorinhibit

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