1. GPCR/G Protein Neuronal Signaling
  2. Adrenergic Receptor
  3. Deriglidole

Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors.

For research use only. We do not sell to patients.

Deriglidole Chemical Structure

Deriglidole Chemical Structure

CAS No. : 122830-14-2

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Description

Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors.

IC50 & Target

Adrenoceptor[1]

In Vitro

Deriglidole is a selective α2-receptor inhibitor. Deriglidole inhibits [3H]Clonidine and [3H]Idazoxan but not [3H]Prazosin binding to rat cortical and human platelet α2-adrenoceptors and is more selective than Idazoxan for peripheral receptors[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

255.36

Formula

C16H21N3

CAS No.
SMILES

CCCC1(C2=NCCN2)N3C4=C(C=CC=C4CC3)C1

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
Deriglidole
Cat. No.:
HY-101683
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