Adrenergic Receptor Inhibitors

α adrenergic receptor

β adrenergic receptor

Adrenergic Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators

Product Name	α adrenergic receptor	β adrenergic receptor	Purity
Isoprenaline hydrochloride		β adrenergic receptor	99.86%
Norepinephrine	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.33%
Zenidolol hydrochloride		β adrenergic receptor	99.76%
Propranolol hydrochloride		β adrenergic receptor	99.97%
Phenylephrine	α adrenergic receptor		99.52%
ORM-10921 free base	Alpha-2C adrenergic receptor, Ki: 1.4 nM
CL 316243		β adrenergic receptor	99.67%
D-Mannitol		Beta-3 adrenergic receptor	99.93%
Phenylephrine hydrochloride	α adrenergic receptor		99.76%
Propranolol		β adrenergic receptor	99.87%
Norepinephrine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.95%
Metoprolol		β1 adrenoceptor	99.89%
Atenolol		Beta-1 adrenergic receptor, Ki: 697 nM	99.94%
Clozapine	α2-adrenergic receptor, Ki: 51 nM (Inhibitor)		99.97%
Prazosin hydrochloride	α adrenergic receptor		99.86%
Norepinephrine bitartrate monohydrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.75%
Dexmedetomidine	α2-adrenergic receptor, Ki: 1.08 nM		99.93%
Mirabegron		β adrenergic receptor	99.90%
Nadolol		β adrenergic receptor	99.97%
Phenylacetylglycine		β2 adrenoceptor	99.63%
Salbutamol		β adrenergic receptor	99.92%
Dexmedetomidine hydrochloride	α2-adrenergic receptor, IC₅₀: 1.08 nM		99.93%
Salmeterol		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.91%
SR59230A		β adrenergic receptor	≥98.0%
Dobutamine hydrochloride	α adrenergic receptor	β adrenergic receptor	99.91%
(S)-Timolol maleate		β adrenergic receptor	99.89%
Vilanterol trifenatate		β adrenergic receptor	99.61%
Labetalol	α1-adrenergic receptor	β-adrenoceptor	99.88%
Guanfacine hydrochloride	α adrenergic receptor		99.96%
L748337		Beta-3 adrenergic receptor, Ki: 4 nM Beta-2 adrenergic receptor, Ki: 204 nM Beta-1 adrenergic receptor, Ki: 390 nM	99.67%
Tamsulosin	α1-adrenergic receptor		99.77%
SR59230A hydrochloride		β adrenergic receptor	99.87%
Phentolamine mesylate	α adrenergic receptor		99.87%
Brimonidine tartrate	α adrenergic receptor		99.14%
Octopamine hydrochloride	α2-adrenergic receptor		99.65%
Paliperidone	α adrenergic receptor		99.69%
Nefazodone hydrochloride	α1-adrenergic receptor		99.87%
Mirtazapine	α2-adrenergic receptor, pKi: 6.95		99.94%
Doxazosin mesylate	α adrenergic receptor		98.34%
Bisoprolol hemifumarate		Beta-1 adrenergic receptor	99.73%
Pronethalol		β adrenergic receptor	99.73%
Atipamezole hydrochloride	α adrenergic receptor		99.97%
Acebutolol hydrochloride		β1 adrenoceptor	99.97%
Fenoterol		β adrenergic receptor	99.25%
Fenoterol hydrobromide		β adrenergic receptor	99.90%
Indacaterol		β adrenergic receptor	99.98%
Salbutamol hemisulfate		β adrenergic receptor	≥98.0%
Indacaterol maleate		β adrenergic receptor	99.81%
Terbutaline sulfate		β adrenergic receptor	99.95%
Vilanterol		β adrenergic receptor	99.30%
Naftopidil	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM		98.47%
Reboxetine mesylate	α adrenergic receptor		99.90%
Metoprolol succinate		β1 adrenoceptor	99.90%
Methyldopa hydrate	α adrenergic receptor		99.95%
Vibegron		β3 adrenoceptor, EC₅₀: 1.1 nM	98.82%
Idazoxan hydrochloride	α adrenergic receptor		99.32%
Medetomidine hydrochloride	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.92%
Midodrine hydrochloride	α adrenergic receptor		99.49%
JP1302 dihydrochloride	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM		99.62%
Lubabegron		β adrenergic receptor	98.21%
Butaxamine hydrochloride		Beta-2 adrenergic receptor	99.87%
Olodaterol		β2 adrenoceptor, EC₅₀: 0.1 nM	98.48%
Asenapine	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5		99.93%
Brimonidine	α adrenergic receptor		99.99%
Salmeterol xinafoate		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.96%
Bufuralol		β-adrenoceptor	99.17%
Blonanserin	α2-adrenergic receptor, Ki: 530 (Rat c nM α1-adrenergic receptor, Ki: 26.7 (Rat nM		99.62%
Ecopipam hydrochloride	Alpha-2A adrenergic receptor, Ki: 731 nM		99.46%
Synephrine		β adrenergic receptor	≥98.0%
Olodaterol hydrochloride		β2 adrenoceptor, EC₅₀: 0.1 nM	98.87%
Harmane	α2-adrenergic receptor, IC₅₀: 18 μM		99.84%
Talipexole dihydrochloride	α2-adrenergic receptor, IC₅₀: 25 nM		99.80%
(S)-(-)-Propranolol hydrochloride		β adrenergic receptor	99.95%
Carazolol		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor	99.71%
Phentolamine	α adrenergic receptor		99.94%
Isoferulic acid	α adrenergic receptor		99.82%
Vatinoxan hydrochloride	α adrenergic receptor		99.89%
LY 344864	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM		98.93%
Medetomidine	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.99%
Levobunolol hydrochloride		β-adrenoceptor	99.89%
Terbutaline		Beta-2 adrenergic receptor	99.65%
Levalbuterol hydrochloride		β adrenergic receptor	99.93%
Bevantolol hydrochloride	α adrenergic receptor	β adrenergic receptor	98.98%
(R)-(+)-Atenolol		β adrenergic receptor	≥99.0%
Oxprenolol hydrochloride		β-adrenoceptor, Ki: 7.1 nM	99.86%
Metipranolol		β1 adrenoceptor, pA2: 8.3 β2 adrenoceptor, pA2: 8.4	98.36%
Isoetharine mesylate		β adrenergic receptor	99.87%
BRL 37344 sodium		β adrenergic receptor	≥99.0%
Xamoterol hemifumarate		β adrenergic receptor	99.92%
Dapiprazole hydrochloride	α1-adrenergic receptor		99.87%
ARC 239 dihydrochloride	Alpha-2B adrenergic receptor		99.57%
CGP 20712 A		β adrenergic receptor	≥99.0%
Bufuralol hydrochloride		β adrenergic receptor	≥99.0%
Xylometazoline hydrochloride	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM		99.58%
(RS)-Butyryltimolol		β adrenergic receptor	≥98.0%
Urapidil hydrochloride	α1-adrenergic receptor, pIC₅₀: 6.13 α2-adrenergic receptor, pIC₅₀: 4.38		99.97%
Synephrine hydrochloride		β adrenergic receptor	99.66%
BMY-14802 hydrochloride	α1-adrenergic receptor		98.02%
Apraclonidine hydrochloride	α adrenergic receptor		98.80%
Clenproperol		β adrenergic receptor	98.26%
Ecopipam hydrobromide	Alpha-2A adrenergic receptor, Ki: 731 nM		≥99.0%
Ajmalicine	α1-adrenergic receptor α2-adrenergic receptor		99.39%
Tasipimidine sulfate	human α2A-adrenoceptor, pEC₅₀: 7.57 rodent α2D-adrenoceptor, pEC₅₀: 6.56 human α2C-adrenoceptor, pEC₅₀: 6.29 human α2B-adrenoceptor, pEC₅₀: 6.00		99.46%
Methyldopate	α adrenergic receptor		98.01%
Tamsulosin hydrochloride	α1-adrenergic receptor		99.81%
A-61603	α1A-adrenergic receptor		≥99.0%
Spiroxatrine	α2-adrenergic receptor		99.18%
Nifenalol hydrochloride		β-adrenoceptor	99.93%
Salmeterol-d₃		β adrenergic receptor	98.91%
NP10679	Alpha-1A adrenergic receptor, IC₅₀: 0.154 μM Alpha-1A adrenergic receptor, Ki: 0.603 μM Alpha-1B adrenergic receptor, Ki: 1.92 μM Alpha-1D adrenergic receptor, Ki: 0.495 μM Alpha-2C adrenergic receptor, Ki: 3.09 μM		99.42%
Scopine hydrochloride	α adrenergic receptor		≥98.0%
Metaterol		β adrenergic receptor
Abanoquil	α1-adrenergic receptor		98.43%
Bupranolol		β-adrenoceptor	99.44%
BMS-466442	α adrenergic receptor, IC₅₀: ≥10 μM		98.99%
Desglymidodrine	α1A-adrenergic receptor, pKi: 5.89 α1B-adrenergic receptor, pKi: 5.16 rat alpha_1D-adrenergic receptor, pKi: 5.78 human α2A-adrenoceptor, pKi: 5.83
Dicentrine	α adrenergic receptor		99.38%
HOKU-81		Beta-2 adrenergic receptor
ST1936	α1-adrenergic receptor, Ki: 390 nM (rat) α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human)		99.70%
Methyldopa	α adrenergic receptor		98.25%
Metoprolol-d₇ hydrochloride		β adrenergic receptor	99.65%
Brombuterol-d₉		β adrenergic receptor	≥99.0%
Mibenratide		Beta-1 adrenergic receptor	99.77%
Higenamine		β adrenergic receptor
Reproterol		β2 adrenoceptor
Efaroxan hydrochloride	α adrenergic receptor		99.94%
Bunazosin	α1-adrenergic receptor		98.52%
Mabuterol		Beta-2 adrenergic receptor	99.96%
Amosulalol	α1-adrenergic receptor	Beta-1 adrenergic receptor	98.69%
BMY 14802	α1-adrenergic receptor		98.96%
Celiprolol hydrochloride		β adrenergic receptor, Ki: 0.14-8.3 μM	98.93%
Xamoterol		β adrenergic receptor
ARC 239	human α2C-adrenoceptor, pKi: 6.95 Alpha-2C adrenergic receptor, pKi: 7.06		99.71%
Prenalterol		β1 adrenoceptor	99.18%
AGN 192836	α adrenergic receptor		99.49%
(Rac)-Rotigotine hydrochloride	Alpha-2B adrenergic receptor		98.66%
CGP 12177 hydrochloride	α1-adrenergic receptor	Beta-1 adrenergic receptor Beta-2 adrenergic receptor Beta-3 adrenergic receptor	99.57%
BMY 7378	rat α_1A-adrenergic receptor, Ki: 800 nM hamster alpha_1B-adrenergic receptor, Ki: 600 nM rat alpha_1D-adrenergic receptor, Ki: 2 nM		99.92%
Midodrine	α adrenergic receptor		99.67%
Metoprolol tartrate		β1 adrenoceptor	99.98%
Isoetharine		β adrenergic receptor
Timolol hemihydrate		β adrenergic receptor
Blonanserin dihydrochloride	α2-adrenergic receptor, Ki: 530 nM α1-adrenergic receptor, Ki: 26.7 nM
Timolol		β adrenergic receptor
(R,R)-Reboxetine mesylate	α adrenergic receptor
Dobutamine	α adrenergic receptor	β adrenergic receptor
Ritodrine		β adrenergic receptor
Metoprolol fumarate		β1 adrenoceptor
Bopindolol fumarate		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor
Trimazosin	α1-adrenergic receptor
Naftopidil dihydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2
RS-79948-197	rat α2A receptor, Kd: 0.42 nM rat α2B recepter, Kd: 0.18 nM rat α2C recepter, Kd: 0.19 nM human α2A-adrenoceptor, Kd: 0.6 nM human α2B-adrenoceptor, Kd: 0.46 nM human α2C-adrenoceptor, Kd: 0.77 nM
Rezatomidine	α2-adrenergic receptor
Amidephrine	α1-adrenergic receptor
Nipradolol	α1-adrenergic receptor
Piribedil dihydrochloride	α adrenergic receptor
Celiprolol		β adrenergic receptor, Ki: 0.14-8.3 μM
Metoprolol-d₆ tartrate		β adrenergic receptor
Zolertine hydrochloride	α1B-adrenergic receptor, pKi: 6.81 (in rat liver membrane) α1A-adrenergic receptor, pKi: 6.35 (in rabbit liver membrane)
SB-206606		Beta-3 adrenergic receptor
Oxprenolol		β-adrenoceptor, Ki: 7.1 nM
Bopindolol		β2 adrenoceptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor
Mabuterol hydrochloride		Beta-2 adrenergic receptor
Nifenalol		Beta-1 adrenergic receptor
Propranolol-d₇ hydrochloride		β adrenergic receptor	98.02%
4-Hydroxypropranolol hydrochloride		β adrenergic receptor
Bisoprolol		Beta-1 adrenergic receptor
(E)-Guanabenz	α adrenergic receptor
ST91	α2-adrenergic receptor		99.75%
α2C adrenoceptor agonist 1	Alpha-2C adrenergic receptor, EC₅₀: 108 nM Alpha-2C adrenergic receptor, Ki: 12 nM
Rec 15/2615 hydrochloride	α1A-adrenergic receptor, Ki: 1.9 nM α1B-adrenergic receptor, Ki: 0.3 nM Alpha-1D adrenergic receptor, Ki: 2.6 nM
Fenoterol hydrobromide (Standard)		β adrenergic receptor
Acebutolol-d₇		β adrenergic receptor
Isamoltane hemifumarate		β-adrenoceptor, IC₅₀: 8.4 nM
Isoprenaline hemisulfate		β adrenergic receptor
S(-)-Bisoprolol fumarate		β adrenergic receptor
Butyryltimolol		β adrenergic receptor	≥98.0%
Butaxamine		β2 adrenoceptor
JP1302	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM
LAS190792		β2 adrenoceptor, pIC₅₀: 9.1 β3 adrenoceptor, pIC₅₀: 5.6 β1 adrenoceptor, pIC₅₀: 7.5
Ajmalicine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor
S(-)-Bisoprolol		β adrenergic receptor
SM-2470	α adrenergic receptor
Acebutolol		β1 adrenoceptor
Bisoprolol fumarate		Beta-1 adrenergic receptor
4-Hydroxypropranolol-d₇ hydrochloride		β adrenergic receptor
DL 071IT		β adrenergic receptor
β2AR/M3-receptor agonist-1		β2 adrenoceptor, pEC₅₀: >9.2
α1A-AR Degrader 9c	α1A-adrenergic receptor, DC₅₀: 2.86 μM
RWJ52353	Alpha-2D adrenergic receptor, Ki: 1.5 nM Alpha-2A adrenergic receptor, Ki: 254 nM α1-adrenergic receptor, Ki: 443 nM Alpha-2B adrenergic receptor, Ki: 621 nM
Naftopidil hydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM
Ecopipam	Alpha-2A adrenergic receptor, Ki: 731 nM
Harmane (Standard)	α2-adrenergic receptor
Diacetolol-d₇		β adrenergic receptor
Mirtazapine (Standard)	α2-adrenergic receptor
Meluadrine		β2 adrenoceptor
ST1936 oxalate	α1-adrenergic receptor, Ki: 390 nM (rat) α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human)
Meluadrine tartrate		β2 adrenoceptor
Cimbuterol-d₉		β adrenergic receptor
SUN-1334H free base	Alpha-1D adrenergic receptor, IC₅₀: 7.76 μM
Dapiprazole	α1-adrenergic receptor
Apraclonidine	α adrenergic receptor
Phenylethanolamine A-d₃		β adrenergic receptor
Moprolol		Beta-1 adrenergic receptor
Pronethalol hydrochloride		β adrenergic receptor
N-5984		β-adrenoceptor
Undecylenoyl phenylalanine		β-adrenoceptor
Asenapine citrate	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5
Metaproterenol		β adrenergic receptor
Levalbuterol		β adrenergic receptor
Clozapine (Standard)	α2-adrenergic receptor		99.98%
BODIPY FL prazosin	α1A-adrenergic receptor, Ki: 14.5 nM α1B-adrenergic receptor, Ki: 43.3 nM
Clenproperol-d₇		β adrenergic receptor
(±)-Penbutolol-d₉ hydrochloride		β adrenergic receptor
Clorprenaline-d₇		β adrenergic receptor
Levobunolol		β adrenergic receptor
2-MPMDQ	α1-adrenergic receptor, Ki: 0.37 nM α2-adrenergic receptor, Ki: 1740 nM
Atenolol (Standard)		Beta-1 adrenergic receptor	99.94%
Sulfinalol		β-adrenoceptor
Mabuterol-d₉		β adrenergic receptor
Agroclavine	α1-adrenergic receptor
Norepinephrine tartrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor
TD-5471 hydrochloride		β adrenergic receptor
Terbutaline sulfate (Standard)		β adrenergic receptor
Methyldopate hydrochloride	α adrenergic receptor
AVN-101 hydrochloride	Alpha-1D adrenergic receptor, Ki: 30.2 nM Alpha-1B adrenergic receptor, Ki: 9.4 nM Alpha-2A adrenergic receptor, Ki: 1.77 nM Alpha-2C adrenergic receptor, Ki: 3.55 nM Alpha-1A adrenergic receptor, Ki: 18.9 nM Alpha-2B adrenergic receptor, Ki: 0.41 nM		99.59%
LY 344864 hydrochloride	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM
β2AR agonist /M-receptor antagonist-1		Beta-2 adrenergic receptor
Brombuterol-d₉ hydrochloride		β adrenergic receptor
CHF-6550		β2 adrenoceptor, pKi: 10.6
Oxyfedrine		β-adrenoceptor
Metrenperone	α1-adrenergic receptor α2-adrenergic receptor
Fluparoxan hydrochloride	α2-adrenergic receptor
Bevantolol		Beta-1 adrenergic receptor
Doxazosin-d₈	α adrenergic receptor
Levobetaxolol		β1 adrenoceptor, IC₅₀: 33.2 nM β2 adrenoceptor, IC₅₀: 2970 nM β3 adrenoceptor, IC₅₀: 709 nM
Todralazine		β adrenergic receptor
Levalbuterol tartrate		β adrenergic receptor
Fluparoxan	α2-adrenergic receptor
Protokylol hydrochloride		Beta-2 adrenergic receptor
Methyldopa hydrochloride	α adrenergic receptor
Xylometazoline	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM
(rac)-Nebivolol-d₄		β adrenergic receptor
Pargolol hydrochloride		β adrenergic receptor
Ko-3290		β adrenergic receptor
Azepexole dihydrochloride	α adrenergic receptor
Clozapine hydrochloride	α2-adrenergic receptor, Ki: 51 nM
Ridazolol		Beta-1 adrenergic receptor
Midaglizole hydrochloride	α adrenergic receptor		99.67%
Benzquinamide	α adrenergic receptor
Fenmetozole Tosylate	α adrenergic receptor

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