2. GPCR/G Protein
  3. GPR4
  4. GPR4 antagonist 1

GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.

For research use only. We do not sell to patients.

GPR4 antagonist 1 Chemical Structure

GPR4 antagonist 1 Chemical Structure

CAS No. : 1197879-16-5

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10 mM * 1 mL in DMSO USD 638 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.

IC50 & Target

IC50: 189 nM (GPR4)[1].
Molecular Weight

431.62

Formula

C27H37N5
CAS No.
Appearance

Oil

Color

Light yellow to yellow

SMILES

CC1=C2C(N(CC3=CC=C(/C=C/CN4CCN(C(C)C)CC4)C=C3)C(CC)=N2)=NC(C)=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation

Purity: 98.92%

COA (245 KB) HNMR (269 KB) LCMS (267 KB)

Handling Instructions (2659 KB)
References
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GPR4 antagonist 1 Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR4 antagonist 11197879-16-5GPR4G Protein-Coupled Receptor 4Inhibitorinhibitorinhibit

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GPR4 antagonist 1
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HY-101536
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