2. PI3K/Akt/mTOR
  3. PI3K
  4. PI3Kγ inhibitor 2

PI3Kγ inhibitor 2 (Compound 16) is an orally bioavailable, CNS-penetrant, isoform selective PI3Kγ inhibitor with a Ki of 4 nM.

For research use only. We do not sell to patients.

PI3Kγ inhibitor 2 Chemical Structure

PI3Kγ inhibitor 2 Chemical Structure

CAS No. : 1315538-79-4

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PI3Kγ inhibitor 2 Related Antibodies

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PI3Kα PI3Kβ PI3Kγ PI3Kδ PI3KC2α PI3KC2β PI3KC2γ Vps34 PI3K PI3KC3 p120γ

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Description

PI3Kγ inhibitor 2 (Compound 16) is an orally bioavailable, CNS-penetrant, isoform selective PI3Kγ inhibitor with a Ki of 4 nM[1].

IC50 & Target[1]

PI3Kγ

4 nM (Ki)

Molecular Weight

433.38

Formula

C20H18F3N5O3
CAS No.
SMILES

O=C1N(C2=CN(CC(F)(F)F)N=C2)[C@H](C)C3=NC(C4=CC(OC)=C(OC)N=C4)=CC=C31
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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PI3Kγ inhibitor 2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PI3Kγ inhibitor 21315538-79-4PI3KPhosphoinositide 3-kinaseInhibitorinhibitorinhibit

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