2. Signaling Pathways
  3. GPCR/G Protein
  4. CRFR
  5. CRFR Inhibitors

CRFR Inhibitors

CRFR1

CRFR2

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

CRFR Inhibitors, Agonists, Antagonists & Modulators
Product Name CRFR1 CRFR2 Purity
R121919
CRFR1, Ki: 2-5 nM
  99.53%
NBI 35965 methanesulfonate
CRFR1, Ki: 4 nM
CRFR1, pKi: 8.5
 
NBI-34041
CRFR1, IC50: 58.9 nM
CRFR1, Ki: 4 nM
CRFR2, IC50: >10000 nM
Cortagine
CRFR1
  99.53%
CP 376395
CRFR1
CRFR2
99.68%
Tildacerfont
CRFR1
  98.25%
Urocortin, rat
CRFR1
CRFR2
α-Helical CRF(9-41) TFA
CRFR1
CRFR2
99.72%
R121919 hydrochloride
CRFR1, Ki: 2-5 nM
 
K41498  
CRFR2
CP 376395 hydrochloride
CRFR1
CRFR2
Urocortin II, human  
CRFR2
NBI 35965 hydrochloride
CRFR1, Ki: 4 nM
CRFR1, pKi: 8.5
 
Urocortin II, mouse
CRFR1, Ki: ﹥100 nM
CRFR2, Ki: 0.66 nM
Urocortin II, human TFA  
CRFR2
(Tyr0)-Urocortin, rat
CRFR1
CRFR2