1. Signaling Pathways
  2. GPCR/G Protein
  3. CaSR
  4. CaSR Modulator

CaSR Modulator

CaSR Modulators (3):

Cat. No. Product Name Effect Purity
  • HY-10167A
    Tecalcet Hydrochloride
    Modulator 99.66%
    Tecalcet Hydrochloride (R 568 Hydrochloride), an orally active calcimimetic compound, allosterically and positively modulates the calcium-sensing receptor (CaSR). Tecalcet Hydrochloride (R 568 Hydrochloride) increases the sensitivity to activation by extracellular Ca2+.
  • HY-112171
    γ-L-Glutamyl-L-alanine
    Modulator ≥98.0%
    γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is a proteolytic breakdown product of larger proteins. γ-L-Glutamyl-L-alanine is a natural substrate of the γ-Glutamylcyclotransferase. γ-L-Glutamyl-L-alanine is a positive modulator of calcium-sensing receptor (CaR) function.
  • HY-10167
    Tecalcet
    Modulator
    Tecalcet (R 568), an orally active calcimimetic compound, allosterically and positively modulates the calcium-sensing receptor (CaSR). Tecalcet (R 568) increases the sensitivity to activation by extracellular Ca2+.