Estrogen Receptor/ERR Agonist

Estrogen Receptor/ERR Agonists (94):

Cat. No.	Product Name	Effect	Purity

HY-132205

DS45500853	Agonist	98.15%
DS45500853 is an estrogen-related receptor α (ERRα) agonist. DS45500853 inhibits the binding between receptor-interacting protein 140 (RIP140) corepressor peptide (10 nM) and GST-ERRα ligand-binding domain (LBD; 1.2 μM) with an IC₅₀ value of 0.80 μM. DS45500853 can be used for the research of metabolic disorders, including type 2 diabetes mellitus (T2DM).

HY-108414

(R)-Equol	Agonist	98.93%
(R)-Equol is an agonist of both ERα and ERβ with K_is of 27.4 and 15.4 nM, respectively.

HY-B1662

Hexestrol	Agonist	99.89%
Hexestrol is a nonsteroidal synthetic estrogen, with a K_i of 0.06 and 0.06 nM for estrogen receptor alpha (ERα) and ERβ. Hexestrol can be used for the research of the diseases caused by estrogen deficiencym, and it also can increase the weight of cattle.

HY-N0322R

Cholesterol (Standard)	Agonist	98.23%
Cholesterol (Standard) is the analytical standard of Cholesterol. This product is intended for research and analytical applications. Cholesterol is the major sterol in mammals. It is making up 20-25% of structural component of the plasma membrane. Plasma membranes are highly permeable to water but relatively impermeable to ions and protons. Cholesterol plays an important role in determining the fluidity and permeability characteristics of the membrane as well as the function of both the transporters and signaling proteins. Cholesterol is also an endogenous estrogen-related receptor α (ERRα) agonist.

HY-101271

WAY-200070	Agonist	99.73%
WAY-200070 is a selective estrogen receptor β (ERβ) agonist with an IC₅₀ of 2.3 nM.

HY-143227

DK3	Agonist	99.82%
DK3 is a potent and selective estrogen-related receptor alpha (ERRα) agonist.

HY-18295

Erteberel	Agonist	99.87%
Erteberel (LY500307) is a potent and selective estrogen receptor beta (ERβ) agonist with K_i and EC₅₀ of 1.54 nM and 3.61 nM, respectively. Erteberel has anti-tumor activities.

HY-B0390

Mestranol	Agonist	99.97%
Mestranol is an inactive proagent and becomes biologically active on conversion to ethinyl estradiol (EE). Mestranol acts as an estrogen receptor agonist. Mestranol combines with a progestin in vivo and can be used for the research of menopausal hormone or menstrual disorders. Mestranol is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

HY-143201

DS20362725	Agonist	99.34%
DS20362725 is an estrogen-related receptor α (ERRα) agonist. DS20362725 inhibits the binding between receptor-interacting protein 140 (RIP140) corepressor peptide (10 nM) and GST-ERRα ligand-binding domain (LBD; 1.2 μM) with an IC₅₀ value of 0.6 μM. DS20362725 can be used for the research of metabolic disorders, including type 2 diabetes mellitus (T2DM).

HY-150210

FSHR agonist 1	Agonist	98.48%
FSHR agonist 1 is a high affinity and allosteric follicle stimulating hormone receptor (FSHR) agonist with a pEC₅₀ of 7.72. FSHR agonist 1 formes extensive interactions with the TMD to directly activate FSHR.

HY-145848

ERRγ agonist-1	Agonist	98.70%
ERRγ agonist-1 is a potent ERRγ agonist. ERRγ agonist-1 increases transcriptional activities of ERRγ. ERRγ agonist-1 has the potential for the research of neuropsychological disorders.

HY-B0708

β-Estradiol 17-acetate	Agonist	99.93%
β-Estradiol 17-acetate is a metabolite of estradiol.

HY-B1012

Quinestrol	Agonist	99.72%
Quinestrol is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

HY-B1403

Dienestrol	Agonist	98.08%
Dienestrol is a synthetic, non-steroidal estrogen, is an estrogen receptor agonist, for the treatment of menopausal and postmenopausal symptoms.

HY-138686

GPR30 agonist-1	Agonist	98.62%
GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects.

HY-B0672R

Estradiol valerate (Standard)	Agonist	99.87%
Estradiol valerianate (Standard) is the analytical standard of Estradiol valerianate. This product is intended for research and analytical applications. Estradiol valerate (β-Estradiol 17-valerate) is a synthetic estrogen widely used in combination with other steroid hormones in hormone replacement therapy agents.

HY-N0322S5

Cholesterol-¹³C₂	Agonist	99.76%
Cholesterol-¹³C₂ is the ¹³C labeled Cholesterol. Cholesterol is the major sterol in mammals. It is making up 20-25% of structural component of the plasma membrane. Plasma membranes are highly permeable to water but relatively impermeable to ions and protons. Cholesterol plays an important role in determining the fluidity and permeability characteristics of the membrane as well as the function of both the transporters and signaling proteins. Cholesterol is also an endogenous estrogen-related receptor α (ERRα) agonist.

HY-B2245

Estradiol dipropionate	Agonist	99.85%
Estradiol dipropionate is a combined estrogen-progesterone, acts as an estrogen and progesterone agonist.

HY-B0234R

Estrone (Standard)	Agonist	99.88%
Estrone (Standard) is the analytical standard of Estrone. This product is intended for research and analytical applications. Estrone (E1) is a natural estrogenic hormone. Estrone is the main representative of the endogenous estrogens and is produced by several tissues, especially adipose tissue. Estrone is the result of the process of aromatization of androstenedione that occurs in fat cells.

HY-B1361

Estropipate	Agonist	98.94%
Estropipate is a form of estrogen, used to treat symptoms of menopause, also used to prevent osteoporosis.

Name
Email *

	Sorry, but the email address you supplied was invalid.