Orexin Receptor (OX Receptor) Inhibitors

OX₂ Receptor

OX₁ Receptor

Orexin Receptor (OX Receptor) Inhibitors, Agonists & Antagonists

Product Name	OX₂ Receptor	OX₁ Receptor	Purity
Orexin A (human, rat, mouse) (acetate)	OX₂ Receptor	OX₁ Receptor	99.93%
Orexin A (human, rat, mouse)	OX₂ Receptor	OX₁ Receptor	99.67%
Almorexant	human OX2R, Kd: 0.17 nM	human OX1R, Kd: 1.3 nM	99.71%
Orexin A (human, rat, mouse) (TFA)	OX₂ Receptor	OX₁ Receptor
OX-201	OX₂ Receptor, EC₅₀: 8 nM	OX₁ Receptor, EC₅₀: 8.1 μM
OX2R-IN-3	OX₂ Receptor, EC₅₀: <100 nM
SB-334867		OX1	99.44%
YNT-185 dihydrochloride	OX₂ Receptor, EC₅₀: 0.028 μM	OX₁ Receptor, EC₅₀: 2.75 μM	99.78%
EMPA	OX₂ Receptor		99.48%
SB-334867 free base	OX2, :	OX₁ Receptor	99.88%
Orexin 2 Receptor Agonist	OX₂ Receptor		99.59%
Seltorexant	human OX2R, pKi: 8.0 rat OX2R, pKi: 8.1		99.86%
SB-674042	OX₂ Receptor, IC₅₀: 531 nM OX₂ Receptor, Ki: 129 nM	OX₁ Receptor, IC₅₀: 3.76 nM OX₁ Receptor, Ki: 1.1 nM	99.93%
MK-1064	OX₂ Receptor, IC₅₀: 18 nM OX₂ Receptor, Ki: 0.5 nM	OX₁ Receptor, IC₅₀: 1789 nM OX₁ Receptor, Ki: 1584 nM	99.95%
OXA(17-33)	OX2, EC₅₀: 187 nM	OX1, EC₅₀: 8.29 nM
TCS-OX2-29	OX₂ Receptor		99.55%
Seltorexant hydrochloride	human OX2R, pKi: 8.0 rat OX2R, pKi: 8.1		99.90%
RTIOXA-43	OX2, EC₅₀: 24 nM	OX1, EC₅₀: 24 nM	99.94%
Almorexant hydrochloride	human OX2R, Kd: 0.17 nM	human OX1R, Kd: 1.3 nM	99.98%
Vornorexant	OX₂ Receptor		99.66%
TCS 1102	OX₂ Receptor, Ki: 0.2 nM	OX₁ Receptor, Ki: 3 nM	99.73%
Firazorexton	OX₂ Receptor		99.94%
GSK1059865		OX₁ Receptor	99.83%
ACT-462206	OX2	OX1	99.60%
SB-408124		OX₁ Receptor, Ki: 57 nM (in whole cell ) OX₁ Receptor, Ki: 27 nM (in cell membrane)	98.27%
ACT-335827	OX2, IC₅₀: 417 nM	OX1, IC₅₀: 6 nM	≥98.0%
[Ala11,D-Leu15]-Orexin B(human)	OX2, EC₅₀: 0.13 nM	OX1, EC₅₀: 52 nM	98.04%
Orexin 2 Receptor Agonist 2	OX₂ Receptor		98.06%
SB-408124 Hydrochloride		OX₁ Receptor, Ki: 57 nM (in whole cell ) OX₁ Receptor, Ki: 27 nM (in cell membrane)	98.79%
TCS-OX2-29 hydrochloride	OX₂ Receptor
CVN766	OX2, IC₅₀: >10 μM	OX1, IC₅₀: 8 nM
[Ala11,D-Leu15]-Orexin B(human) TFA	OX2, EC₅₀: 0.13	OX1, EC₅₀: 52
Hypocretin (70-98), human		human OX1R
OXA(17-33) TFA	OX2, EC₅₀: 187 nM	OX1, EC₅₀: 8.29 nM
Orexin receptor antagonist 4	OX₂ Receptor, IC₅₀: 4.27 nM	OX₁ Receptor, IC₅₀: 295 nM
Almorexant-¹³C,d₃	OX₂ Receptor
OX2R-IN-1	OX₂ Receptor
OX2R-IN-2	OX₂ Receptor, EC₅₀: 339 nM
JNJ-54717793	human OX2R, Ki: 700 nM	human OX1R, Ki: 16 nM OX₁ Receptor, EC₅₀: 85 ng/mL	98.85%
MK-8133	OX₂ Receptor

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