1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. SGLT
  4. SGLT Inhibitors

SGLT Inhibitors

SGLT1

SGLT2

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Please try each isoform separately.

SGLT Inhibitors
Product Name SGLT1 SGLT2 Purity
Dapagliflozin  
SGLT2
99.97%
Canagliflozin  
SGLT2
99.80%
Phloretin
SGLT1
SGLT2
99.67%
SGLT2-IN-1  
SGLT2, IC50: 33 nM
≥98.0%
Atigliflozin
hSGLT1, IC50: 8.2 μM
hSGLT2, IC50: 10 nM
Ertugliflozin  
SGLT2
99.92%
Phlorizin
SGLT1
SGLT2
99.93%
Mizagliflozin
SGLT1
  98.87%
Ipragliflozin
hSGLT1, IC50: 1876 nM
rSGLT1, IC50: 1166 nM
mSGLT1, IC50: 1380 nM
hSGLT2, IC50: 7.38 nM
rSGLT2, IC50: 6.73 nM
mSGLT2, IC50: 5.64 nM
99.78%
Dapagliflozin ((2S)-1,2-propanediol, hydrate)  
SGLT2
99.99%
Canagliflozin hemihydrate  
SGLT2
99.95%
Trilobatin
SGLT1
SGLT2
99.00%
Remogliflozin etabonate
hSGLT1, Ki: 43.1 μM
rSGLT1, Ki: 8.57 μM
hSGLT2, Ki: 1.95 μM
rSGLT2, Ki: 2.14 μM
99.81%
Velagliflozin  
SGLT2
99.92%
Dapagliflozin-d5  
SGLT2
98.01%
Ertugliflozin L-pyroglutamic acid  
SGLT2
99.84%
Enavogliflozin  
SGLT2
98.01%
Ipragliflozin L-Proline  
SGLT2
99.94%
Canagliflozin-d4  
SGLT2
99.04%
Remogliflozin  
SGLT2
SGLT1/2-IN-1
SGLT1, IC50: 15.72 mM
SGLT2, IC50: 3.67 mM
LX2761
SGLT1
SGLT2
Luseogliflozin hydrate  
SGLT2
Luseogliflozin
SGLT1, IC50: 3990 nM
SGLT2, IC50: 2.26 nM
99.20%
Phloretin (Standard)
SGLT1
SGLT2
Sergliflozin etabonate  
SGLT2
Kushenol K
SGLT1
SGLT2
T-1095
hSGLT1, IC50: 22.8 μM
hSGLT2, IC50: 2.3 μM
Velagliflozin proline hydrate  
SGLT2
99.43%
TA-1887
SGLT1, IC50: 230 nM
SGLT2, IC50: 1.4 nM
YM543 free base  
SGLT2
galacto-Dapagliflozin
hSGLT1, Ki: 25000 nM
hSGLT2, Ki: 25 nM
fluoro-Dapagliflozin
hSGLT1, Ki: 330 nM
hSGLT2, Ki: 5.3 nM