2. Metabolic Enzyme/Protease Vitamin D Related/Nuclear Receptor Cell Cycle/DNA Damage Epigenetics PI3K/Akt/mTOR
  3. Adiponectin Receptor PPAR PGC-1α Sirtuin AMPK
  4. AdipoR agonist 1

AdipoR agonist 1 (Compound 112254) is an agonist for adiponectin receptor (AdipoR), which activates the transcriptional regulators like peroxisome proliferator-activated receptors (PPARs), peroxisome proliferator-activated receptor gamma coactivator 1α (PGC-1α), sirtuin 1 (SIRT1), and adenylate-activated protein kinase (AMPK). AdipoR agonist 1 is utilized in preventive doping research.

For research use only. We do not sell to patients.

AdipoR agonist 1 Chemical Structure

AdipoR agonist 1 Chemical Structure

CAS No. : 949745-75-9

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AdipoR agonist 1 Related Antibodies

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NUAK1 NUAK2 AMPK AMPK α1β1γ1 AMPK α2β1γ1 AMPK α1β2γ1 AMPK α2β2γ1

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Description

AdipoR agonist 1 (Compound 112254) is an agonist for adiponectin receptor (AdipoR), which activates the transcriptional regulators like peroxisome proliferator-activated receptors (PPARs), peroxisome proliferator-activated receptor gamma coactivator 1α (PGC-1α), sirtuin 1 (SIRT1), and adenylate-activated protein kinase (AMPK). AdipoR agonist 1 is utilized in preventive doping research[1].

Molecular Weight

437.57

Formula

C26H35N3O3
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(NCCC(N1CCN(CC2=CC=C(OC)C=C2)CC1)=O)C3=CC=C(C(C)(C)C)C=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 5 mg/mL (11.43 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2853 mL 11.4267 mL 22.8535 mL
5 mM 0.4571 mL 2.2853 mL 4.5707 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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This equation is commonly abbreviated as: C1V1 = C2V2

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Working solution concentration: mg/mL
Purity & Documentation

Purity: ≥98.0%

SDS (393 KB)

COA (242 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.2853 mL 11.4267 mL 22.8535 mL 57.1337 mL
5 mM 0.4571 mL 2.2853 mL 4.5707 mL 11.4267 mL
10 mM 0.2285 mL 1.1427 mL 2.2853 mL 5.7134 mL
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AdipoR agonist 1 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

AdipoR agonist 1949745-75-9AdipoR agonist1AdipoR agonist-1Adiponectin ReceptorPPARPGC-1αSirtuinAMPKAdipoRsPeroxisome proliferator-activated receptorsPPARγ coactivator-1αAMP-activated protein kinaseSprague Dawley ratdopingInhibitorinhibitorinhibit

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