2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Azepexole hydrochloride

Azepexole hydrochloride  (Synonyms: B-HT 933 hydrochloride; Oxazoloazepin hydrochloride)

Cat. No.: HY-103212A
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Azepexole hydrochloride (B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride) is a selective agonist for α 2-adrenoceptor, with pKi of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions with IC50 of 78.72 nM. Azepexole hydrochloride exhibits antitussive and analgesic efficacy.

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Azepexole hydrochloride Chemical Structure

Azepexole hydrochloride Chemical Structure

CAS No. : 147663-20-5

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Azepexole hydrochloride Related Antibodies

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Description

Azepexole hydrochloride (B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride) is a selective agonist for α 2-adrenoceptor, with pKi of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions with IC50 of 78.72 nM. Azepexole hydrochloride exhibits antitussive and analgesic efficacy[1][2].

Molecular Weight

217.70

Formula

C9H16ClN3O
CAS No.
SMILES

CCN(CC1)CCC2=C1OC(N)=N2.Cl
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
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Azepexole hydrochloride Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Azepexole147663-20-5B-HT 933OxazoloazepinAdrenergic ReceptorBeta Receptorvasopressorresponsesdiabeticperistaltic contractionsInhibitorinhibitorinhibit

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