1. GPCR/G Protein Neuronal Signaling
  2. Adrenergic Receptor
  3. Azepexole hydrochloride

Azepexole hydrochloride  (Synonyms: B-HT 933 hydrochloride; Oxazoloazepin hydrochloride)

Cat. No.: HY-103212A
Handling Instructions

Azepexole hydrochloride (B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride) is a selective agonist for α 2-adrenoceptor, with pKi of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions with IC50 of 78.72 nM. Azepexole hydrochloride exhibits antitussive and analgesic efficacy.

For research use only. We do not sell to patients.

Azepexole hydrochloride Chemical Structure

Azepexole hydrochloride Chemical Structure

CAS No. : 147663-20-5

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Description

Azepexole hydrochloride (B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride) is a selective agonist for α 2-adrenoceptor, with pKi of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions with IC50 of 78.72 nM. Azepexole hydrochloride exhibits antitussive and analgesic efficacy[1][2].

Molecular Weight

217.70

Formula

C9H16ClN3O

CAS No.
SMILES

CCN(CC1)CCC2=C1OC(N)=N2.Cl

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
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Azepexole hydrochloride Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
Azepexole hydrochloride
Cat. No.:
HY-103212A
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